Targeting topoisomerase I cleavage to specific sequences of DNA by triple helix-forming oligonucleotide conjugates. A comparison between a rebeccamycin derivative and camptothecin.

Arimondo, P B

Targeting topoisomerase I cleavage to specific sequences of DNA by triple helix-forming oligonucleotide conjugates. A comparison between a rebeccamycin derivative and camptothecin. [electronic resource] - Comptes rendus de l'Academie des sciences. Serie III, Sciences de la vie Sep 1999 - 785-90 p. digital

Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't

0764-4469

10.1016/s0764-4469(00)80037-2 doi


Aminoglycosides
Anti-Bacterial Agents--chemistry
Antineoplastic Agents--chemistry
Base Sequence
Camptothecin--chemistry
DNA Topoisomerases, Type I--metabolism
Drug Design
Enzyme Inhibitors--pharmacology
Humans
Molecular Sequence Data
Nucleic Acid Conformation
Oligodeoxyribonucleotides--chemistry
Substrate Specificity
Topoisomerase I Inhibitors