Cardiovascular characterization of pyrrolo[2,1-d][1,5]benzothiazepine derivatives binding selectively to the peripheral-type benzodiazepine receptor (PBR): from dual PBR affinity and calcium antagonist activity to novel and selective calcium entry blockers. [electronic resource]
Producer: 19960906Description: 2922-38 p. digitalISSN:- 0022-2623
- Animals
- Atrial Function
- Binding, Competitive
- Calcium Channel Blockers -- chemical synthesis
- Calcium Channels -- metabolism
- Cardiovascular System -- drug effects
- Cerebral Cortex -- metabolism
- Depression, Chemical
- Female
- Guinea Pigs
- Heart Rate -- drug effects
- Male
- Models, Molecular
- Myocardial Contraction -- drug effects
- Myocardium -- metabolism
- Pyrroles -- chemical synthesis
- Rats
- Rats, Sprague-Dawley
- Receptors, GABA-A -- metabolism
- Structure-Activity Relationship
- Thiazepines -- chemical synthesis
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Publication Type: Comparative Study; Journal Article; Research Support, Non-U.S. Gov't
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