Intrinsic activity and effects of guanyl-5'-yl imidodiphosphate, Gpp(NH)p and sodium ion on the affinity of dynorphin 1-13, nalorphine and nalorphine-7,8-oxide to kappa-opioid receptor. [electronic resource]
Producer: 19860312Description: 617-9 p. digitalISSN:- 0306-3623
- Animals
- Binding, Competitive -- drug effects
- Brain -- metabolism
- Cyclazocine -- analogs & derivatives
- Dynorphins -- antagonists & inhibitors
- Ethylketocyclazocine
- Guanosine Triphosphate -- analogs & derivatives
- Guanylyl Imidodiphosphate -- pharmacology
- In Vitro Techniques
- Male
- Mice
- Mice, Inbred Strains
- Muscle Contraction -- drug effects
- Muscle, Smooth -- drug effects
- Nalorphine -- analogs & derivatives
- Naloxone -- antagonists & inhibitors
- Peptide Fragments -- antagonists & inhibitors
- Rats
- Receptors, Opioid -- drug effects
- Receptors, Opioid, kappa
- Sodium -- pharmacology
- Synaptosomes -- metabolism
- Vas Deferens -- drug effects
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Publication Type: Journal Article
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