Intrinsic activity and effects of guanyl-5'-yl imidodiphosphate, Gpp(NH)p and sodium ion on the affinity of dynorphin 1-13, nalorphine and nalorphine-7,8-oxide to kappa-opioid receptor.

Takayanagi, I

Intrinsic activity and effects of guanyl-5'-yl imidodiphosphate, Gpp(NH)p and sodium ion on the affinity of dynorphin 1-13, nalorphine and nalorphine-7,8-oxide to kappa-opioid receptor. [electronic resource] - General pharmacology 1985 - 617-9 p. digital

Publication Type: Journal Article

0306-3623

10.1016/0306-3623(85)90153-3 doi


Animals
Binding, Competitive--drug effects
Brain--metabolism
Cyclazocine--analogs & derivatives
Dynorphins--antagonists & inhibitors
Ethylketocyclazocine
Guanosine Triphosphate--analogs & derivatives
Guanylyl Imidodiphosphate--pharmacology
In Vitro Techniques
Male
Mice
Mice, Inbred Strains
Muscle Contraction--drug effects
Muscle, Smooth--drug effects
Nalorphine--analogs & derivatives
Naloxone--antagonists & inhibitors
Peptide Fragments--antagonists & inhibitors
Rats
Receptors, Opioid--drug effects
Receptors, Opioid, kappa
Sodium--pharmacology
Synaptosomes--metabolism
Vas Deferens--drug effects