Structural Basis of Transcription Inhibition by CBR Hydroxamidines and CBR Pyrazoles. [electronic resource]
Producer: 20160520Description: 1470-1481 p. digitalISSN:- 1878-4186
- Amidines -- chemistry
- Amino Acid Sequence
- Animals
- Anti-Bacterial Agents -- chemistry
- Binding Sites
- Chlorocebus aethiops
- Crystallography, X-Ray
- DNA-Directed RNA Polymerases -- antagonists & inhibitors
- Drug Synergism
- Escherichia coli -- drug effects
- Escherichia coli Proteins -- antagonists & inhibitors
- HeLa Cells
- Humans
- Hydroxylamines -- chemistry
- Ligands
- Models, Molecular
- Molecular Sequence Data
- Mycobacterium tuberculosis -- drug effects
- Protein Binding
- Protein Structure, Secondary
- Protein Structure, Tertiary
- Pyrazoles -- chemistry
- Recombinant Proteins -- chemistry
- Sequence Alignment
- Transcription, Genetic -- drug effects
- Vero Cells
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Publication Type: Journal Article; Research Support, N.I.H., Extramural
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