Structural Basis of Transcription Inhibition by CBR Hydroxamidines and CBR Pyrazoles.

Feng, Yu

Structural Basis of Transcription Inhibition by CBR Hydroxamidines and CBR Pyrazoles. [electronic resource] - Structure (London, England : 1993) Aug 2015 - 1470-1481 p. digital

Publication Type: Journal Article; Research Support, N.I.H., Extramural

1878-4186

10.1016/j.str.2015.06.009 doi


Amidines--chemistry
Amino Acid Sequence
Animals
Anti-Bacterial Agents--chemistry
Binding Sites
Chlorocebus aethiops
Crystallography, X-Ray
DNA-Directed RNA Polymerases--antagonists & inhibitors
Drug Synergism
Escherichia coli--drug effects
Escherichia coli Proteins--antagonists & inhibitors
HeLa Cells
Humans
Hydroxylamines--chemistry
Ligands
Models, Molecular
Molecular Sequence Data
Mycobacterium tuberculosis--drug effects
Protein Binding
Protein Structure, Secondary
Protein Structure, Tertiary
Pyrazoles--chemistry
Recombinant Proteins--chemistry
Sequence Alignment
Transcription, Genetic--drug effects
Vero Cells