Early rapid identification of in vivo rat metabolites of AN6414, a novel boron-containing PDE4 inhibitor by QTRAP LC/MS/MS to support drug discovery. [electronic resource]
Producer: 20130207Description: 344-53 p. digitalISSN:- 1873-264X
- Administration, Oral
- Animals
- Anti-Inflammatory Agents -- administration & dosage
- Area Under Curve
- Biotransformation
- Boron Compounds -- administration & dosage
- Chromatography, Liquid
- Drug Discovery -- methods
- Female
- Male
- Metabolic Clearance Rate
- Models, Biological
- Oxidation-Reduction
- Phosphodiesterase 4 Inhibitors -- administration & dosage
- Pyridines -- administration & dosage
- Rats
- Rats, Sprague-Dawley
- Risk Assessment
- Software
- Solid Phase Extraction
- Sulfates -- pharmacokinetics
- Tandem Mass Spectrometry
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Publication Type: Journal Article
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