Glucuronidation and covalent protein binding of benoxaprofen and flunoxaprofen in sandwich-cultured rat and human hepatocytes. [electronic resource]
Producer: 20100126Description: 2314-22 p. digitalISSN:- 1521-009X
- Adult
- Animals
- Anti-Inflammatory Agents, Non-Steroidal -- metabolism
- Benzoxazoles -- metabolism
- Biotransformation
- Cell Culture Techniques
- Collagen
- Dose-Response Relationship, Drug
- Drug Combinations
- Feasibility Studies
- Glucuronates -- metabolism
- Glucuronosyltransferase -- metabolism
- Hepatocytes -- metabolism
- Humans
- Ibuprofen -- metabolism
- Kinetics
- Laminin
- Male
- Microsomes, Liver -- metabolism
- Models, Biological
- Propionates -- metabolism
- Protein Binding
- Proteoglycans
- Rats
- Rats, Sprague-Dawley
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Publication Type: Comparative Study; Journal Article; Research Support, N.I.H., Extramural
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