Nicotine is a selective pharmacological chaperone of acetylcholine receptor number and stoichiometry. Implications for drug discovery. [electronic resource]
Producer: 20090723Description: 167-77 p. digitalISSN:- 1550-7416
- Acetylcholine -- metabolism
- Animals
- Drug Discovery
- Endoplasmic Reticulum -- drug effects
- Epilepsy, Frontal Lobe -- genetics
- Hippocampus -- drug effects
- Mice
- Models, Biological
- Muscle Proteins -- biosynthesis
- Mutation, Missense
- Nerve Tissue Proteins -- biosynthesis
- Neurotransmitter Agents -- physiology
- Nicotine -- pharmacokinetics
- Parkinson Disease -- prevention & control
- Receptors, Nicotinic -- biosynthesis
- Smoking -- metabolism
- Tobacco Use Disorder -- genetics
- Up-Regulation -- drug effects
- Ventral Tegmental Area -- drug effects
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Publication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't; Review
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