Replacement of histidine in position 105 in the α₅ subunit by cysteine stimulates zolpidem sensitivity of α₅β₂γ₂ GABA(A) receptors. [electronic resource]
Producer: 20110719Description: 2556-64 p. digitalISSN:- 1471-4159
- Amino Acid Substitution -- physiology
- Animals
- Cysteine -- physiology
- Dose-Response Relationship, Drug
- Electrophysiological Phenomena
- Excitatory Amino Acid Agonists -- pharmacology
- GABA Agonists -- pharmacology
- Histidine -- physiology
- Humans
- Hydrogen-Ion Concentration
- Oocytes -- metabolism
- Patch-Clamp Techniques
- Pyridines -- pharmacology
- Receptors, GABA-A -- drug effects
- Structure-Activity Relationship
- Xenopus
- Zolpidem
- gamma-Aminobutyric Acid -- pharmacology
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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