The high affinity peripheral benzodiazepine receptor ligand DAA1106 binds to activated and infected brain macrophages in areas of synaptic degeneration: implications for PET imaging of neuroinflammation in lentiviral encephalitis. [electronic resource]
Producer: 20080404Description: 232-41 p. digitalISSN:- 0969-9961
- Acetamides -- pharmacokinetics
- Adult
- Aged
- Analysis of Variance
- Animals
- Antigens, CD -- metabolism
- Antigens, Differentiation, Myelomonocytic -- metabolism
- Astrocytes -- drug effects
- Brain -- diagnostic imaging
- Bucladesine -- pharmacology
- Dose-Response Relationship, Drug
- Encephalitis, Viral -- pathology
- Female
- Humans
- Lentivirus
- Lipopolysaccharides -- pharmacology
- Macaca mulatta
- Macrophages -- drug effects
- Male
- Middle Aged
- Nerve Tissue Proteins -- metabolism
- Phenyl Ethers -- pharmacokinetics
- Positron-Emission Tomography
- Protein Binding -- drug effects
- Synapses -- drug effects
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Publication Type: Journal Article; Research Support, N.I.H., Extramural
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