N-desmethylclozapine, an allosteric agonist at muscarinic 1 receptor, potentiates N-methyl-D-aspartate receptor activity. [electronic resource]
Producer: 20040105Description: 13674-9 p. digitalISSN:- 0027-8424
- Allosteric Site
- Animals
- Brain -- metabolism
- Cell Line
- Clozapine -- analogs & derivatives
- Cricetinae
- DNA, Complementary -- metabolism
- Dose-Response Relationship, Drug
- Electrophysiology
- Guanosine 5'-O-(3-Thiotriphosphate) -- metabolism
- Hippocampus -- metabolism
- Humans
- Inhibitory Concentration 50
- Mutagenesis, Site-Directed
- Neurons -- metabolism
- Protein Binding
- Rats
- Receptor, Muscarinic M1 -- agonists
- Receptors, N-Methyl-D-Aspartate -- metabolism
- Time Factors
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Publication Type: Journal Article
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