N-desmethylclozapine, an allosteric agonist at muscarinic 1 receptor, potentiates N-methyl-D-aspartate receptor activity.
Sur, Cyrille
N-desmethylclozapine, an allosteric agonist at muscarinic 1 receptor, potentiates N-methyl-D-aspartate receptor activity. [electronic resource] - Proceedings of the National Academy of Sciences of the United States of America Nov 2003 - 13674-9 p. digital
Publication Type: Journal Article
0027-8424
10.1073/pnas.1835612100 doi
Allosteric Site
Animals
Brain--metabolism
Cell Line
Clozapine--analogs & derivatives
Cricetinae
DNA, Complementary--metabolism
Dose-Response Relationship, Drug
Electrophysiology
Guanosine 5'-O-(3-Thiotriphosphate)--metabolism
Hippocampus--metabolism
Humans
Inhibitory Concentration 50
Mutagenesis, Site-Directed
Neurons--metabolism
Protein Binding
Rats
Receptor, Muscarinic M1--agonists
Receptors, N-Methyl-D-Aspartate--metabolism
Time Factors
N-desmethylclozapine, an allosteric agonist at muscarinic 1 receptor, potentiates N-methyl-D-aspartate receptor activity. [electronic resource] - Proceedings of the National Academy of Sciences of the United States of America Nov 2003 - 13674-9 p. digital
Publication Type: Journal Article
0027-8424
10.1073/pnas.1835612100 doi
Allosteric Site
Animals
Brain--metabolism
Cell Line
Clozapine--analogs & derivatives
Cricetinae
DNA, Complementary--metabolism
Dose-Response Relationship, Drug
Electrophysiology
Guanosine 5'-O-(3-Thiotriphosphate)--metabolism
Hippocampus--metabolism
Humans
Inhibitory Concentration 50
Mutagenesis, Site-Directed
Neurons--metabolism
Protein Binding
Rats
Receptor, Muscarinic M1--agonists
Receptors, N-Methyl-D-Aspartate--metabolism
Time Factors