Inhibitory potencies of 1,4-dihydropyridine calcium antagonists to P-glycoprotein-mediated transport: comparison with the effects on CYP3A4. [electronic resource]
Producer: 20010301Description: 1189-97 p. digitalISSN:- 0724-8741
- ATP Binding Cassette Transporter, Subfamily B, Member 1 -- antagonists & inhibitors
- Animals
- Biological Transport -- drug effects
- Calcium Channel Blockers -- pharmacology
- Cell Line
- Cytochrome P-450 CYP3A
- Cytochrome P-450 Enzyme Inhibitors
- Cytochrome P-450 Enzyme System -- metabolism
- Daunorubicin -- pharmacokinetics
- Digoxin -- pharmacokinetics
- Dihydropyridines -- pharmacology
- Humans
- Mixed Function Oxygenases -- antagonists & inhibitors
- Substrate Specificity
- Transfection
- Tritium
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Publication Type: Comparative Study; Journal Article
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