Inhibitory potencies of 1,4-dihydropyridine calcium antagonists to P-glycoprotein-mediated transport: comparison with the effects on CYP3A4.

Katoh, M

Inhibitory potencies of 1,4-dihydropyridine calcium antagonists to P-glycoprotein-mediated transport: comparison with the effects on CYP3A4. [electronic resource] - Pharmaceutical research Oct 2000 - 1189-97 p. digital

Publication Type: Comparative Study; Journal Article

0724-8741

10.1023/a:1007568811691 doi


ATP Binding Cassette Transporter, Subfamily B, Member 1--antagonists & inhibitors
Animals
Biological Transport--drug effects
Calcium Channel Blockers--pharmacology
Cell Line
Cytochrome P-450 CYP3A
Cytochrome P-450 Enzyme Inhibitors
Cytochrome P-450 Enzyme System--metabolism
Daunorubicin--pharmacokinetics
Digoxin--pharmacokinetics
Dihydropyridines--pharmacology
Humans
Mixed Function Oxygenases--antagonists & inhibitors
Substrate Specificity
Transfection
Tritium