| 000 | 01556 a2200421 4500 | ||
|---|---|---|---|
| 005 | 20250518101418.0 | ||
| 264 | 0 | _c20210614 | |
| 008 | 202106s 0 0 eng d | ||
| 022 | _a1860-7187 | ||
| 024 | 7 |
_a10.1002/cmdc.202000150 _2doi |
|
| 040 |
_aNLM _beng _cNLM |
||
| 100 | 1 | _aAsquith, Christopher R M | |
| 245 | 0 | 0 |
_aTargeting the Water Network in Cyclin G-Associated Kinase (GAK) with 4-Anilino-quin(az)oline Inhibitors. _h[electronic resource] |
| 260 |
_bChemMedChem _c07 2020 |
||
| 300 |
_a1200-1215 p. _bdigital |
||
| 500 | _aPublication Type: Journal Article; Research Support, Non-U.S. Gov't | ||
| 650 | 0 | 4 | _aCrystallography, X-Ray |
| 650 | 0 | 4 | _aDose-Response Relationship, Drug |
| 650 | 0 | 4 | _aHEK293 Cells |
| 650 | 0 | 4 | _aHumans |
| 650 | 0 | 4 |
_aIntracellular Signaling Peptides and Proteins _xantagonists & inhibitors |
| 650 | 0 | 4 | _aModels, Molecular |
| 650 | 0 | 4 | _aMolecular Structure |
| 650 | 0 | 4 |
_aProtein Kinase Inhibitors _xchemical synthesis |
| 650 | 0 | 4 |
_aProtein Serine-Threonine Kinases _xantagonists & inhibitors |
| 650 | 0 | 4 |
_aQuinazolines _xchemical synthesis |
| 650 | 0 | 4 | _aStructure-Activity Relationship |
| 650 | 0 | 4 |
_aWater _xchemistry |
| 700 | 1 | _aTizzard, Graham J | |
| 700 | 1 | _aBennett, James M | |
| 700 | 1 | _aWells, Carrow I | |
| 700 | 1 | _aElkins, Jonathan M | |
| 700 | 1 | _aWillson, Timothy M | |
| 700 | 1 | _aPoso, Antti | |
| 700 | 1 | _aLaitinen, Tuomo | |
| 773 | 0 |
_tChemMedChem _gvol. 15 _gno. 13 _gp. 1200-1215 |
|
| 856 | 4 | 0 |
_uhttps://doi.org/10.1002/cmdc.202000150 _zAvailable from publisher's website |
| 999 |
_c30924511 _d30924511 |
||