000 01695 a2200457 4500
005 20250518093332.0
264 0 _c20201214
008 202012s 0 0 eng d
022 _a1873-2968
024 7 _a10.1016/j.bcp.2020.113938
_2doi
040 _aNLM
_beng
_cNLM
100 1 _aOrtega Ugalde, Sandra
245 0 0 _aAcetylene containing cyclo(L-Tyr-L-Tyr)-analogs as mechanism-based inhibitors of CYP121A1 from Mycobacterium tuberculosis.
_h[electronic resource]
260 _bBiochemical pharmacology
_c07 2020
300 _a113938 p.
_bdigital
500 _aPublication Type: Journal Article; Research Support, Non-U.S. Gov't
650 0 4 _aAcetylene
_xchemistry
650 0 4 _aAntitubercular Agents
_xchemistry
650 0 4 _aCatalytic Domain
650 0 4 _aCyclization
650 0 4 _aCytochrome P-450 Enzyme Inhibitors
_xchemistry
650 0 4 _aCytochrome P-450 Enzyme System
_xchemistry
650 0 4 _aDiketopiperazines
_xmetabolism
650 0 4 _aDipeptides
_xchemistry
650 0 4 _aDrug Design
650 0 4 _aEscherichia coli
_xgenetics
650 0 4 _aMicrobial Sensitivity Tests
650 0 4 _aMycobacterium tuberculosis
_xdrug effects
650 0 4 _aOxidation-Reduction
650 0 4 _aPeptides, Cyclic
_xchemistry
650 0 4 _aSubstrate Specificity
650 0 4 _aTuberculosis
_xmetabolism
650 0 4 _aTyrosine
_xanalogs & derivatives
700 1 _aWallraven, Kerstin
700 1 _aSpeer, Alexander
700 1 _aBitter, Wilbert
700 1 _aGrossmann, Tom N
700 1 _aCommandeur, Jan N M
773 0 _tBiochemical pharmacology
_gvol. 177
_gp. 113938
856 4 0 _uhttps://doi.org/10.1016/j.bcp.2020.113938
_zAvailable from publisher's website
999 _c30792012
_d30792012