000 01979 a2200625 4500
005 20250517211645.0
264 0 _c20181227
008 201812s 0 0 eng d
022 _a1464-3405
024 7 _a10.1016/j.bmcl.2018.04.002
_2doi
040 _aNLM
_beng
_cNLM
100 1 _aMou, Jianfeng
245 0 0 _aStructure-activity relationship study of a series of caspase inhibitors containing γ-amino acid moiety for treatment of cholestatic liver disease.
_h[electronic resource]
260 _bBioorganic & medicinal chemistry letters
_c06 2018
300 _a1874-1878 p.
_bdigital
500 _aPublication Type: Journal Article
650 0 4 _aAmino Acids
_xchemistry
650 0 4 _aAnimals
650 0 4 _aBilirubin
_xblood
650 0 4 _aBinding Sites
650 0 4 _aCaspase 1
_xchemistry
650 0 4 _aCaspase Inhibitors
_xchemistry
650 0 4 _aDisease Models, Animal
650 0 4 _aHalf-Life
650 0 4 _aHumans
650 0 4 _aJurkat Cells
650 0 4 _aLiver Diseases
_xdrug therapy
650 0 4 _aMice
650 0 4 _aMolecular Docking Simulation
650 0 4 _aProtein Structure, Tertiary
650 0 4 _aStructure-Activity Relationship
650 0 4 _afas Receptor
_xantagonists & inhibitors
700 1 _aWu, Songliang
700 1 _aLuo, Zhi
700 1 _aGuo, Fengying
700 1 _aHe, Haiying
700 1 _aWang, Jianhua
700 1 _aLin, Fusen
700 1 _aGuo, Fengxun
700 1 _aSun, Jianping
700 1 _aShen, Liang
700 1 _aZeng, Minggao
700 1 _aWang, Chuan
700 1 _aXu, Deming
700 1 _aGu, Zhengxian
700 1 _aTian, Xin
700 1 _aZhang, Aiming
700 1 _aXu, Hongjiang
700 1 _aYang, Ling
700 1 _aZhang, Xiquan
700 1 _aLi, Jian
700 1 _aChen, Shuhui
773 0 _tBioorganic & medicinal chemistry letters
_gvol. 28
_gno. 10
_gp. 1874-1878
856 4 0 _uhttps://doi.org/10.1016/j.bmcl.2018.04.002
_zAvailable from publisher's website
999 _c28282349
_d28282349