000 01909 a2200553 4500
005 20250517165510.0
264 0 _c20170908
008 201709s 0 0 eng d
022 _a1464-3405
024 7 _a10.1016/j.bmcl.2017.07.052
_2doi
040 _aNLM
_beng
_cNLM
100 1 _aDing, Xiao
245 0 0 _aDiscovery of 5-substituent-N-arylbenzamide derivatives as potent, selective and orally bioavailable LRRK2 inhibitors.
_h[electronic resource]
260 _bBioorganic & medicinal chemistry letters
_c09 2017
300 _a4034-4038 p.
_bdigital
500 _aPublication Type: Journal Article; Research Support, Non-U.S. Gov't
650 0 4 _aAdministration, Oral
650 0 4 _aBenzamides
_xadministration & dosage
650 0 4 _aDose-Response Relationship, Drug
650 0 4 _aDrug Discovery
650 0 4 _aHumans
650 0 4 _aLeucine-Rich Repeat Serine-Threonine Protein Kinase-2
_xantagonists & inhibitors
650 0 4 _aMolecular Structure
650 0 4 _aProtein Kinase Inhibitors
_xadministration & dosage
650 0 4 _aStructure-Activity Relationship
700 1 _aDai, Xuedong
700 1 _aLong, Kai
700 1 _aPeng, Cheng
700 1 _aAndreotti, Daniele
700 1 _aBamborough, Paul
700 1 _aEatherton, Andrew J
700 1 _aEdge, Colin
700 1 _aJandu, Karamjit S
700 1 _aNichols, Paula L
700 1 _aPhilps, Oliver J
700 1 _aStasi, Luigi Piero
700 1 _aWan, Zehong
700 1 _aXiang, Jia-Ning
700 1 _aDong, Kelly
700 1 _aDossang, Pamela
700 1 _aHo, Ming-Hsun
700 1 _aLi, Yi
700 1 _aMensah, Lucy
700 1 _aGuan, Xiaoming
700 1 _aReith, Alastair D
700 1 _aRen, Feng
773 0 _tBioorganic & medicinal chemistry letters
_gvol. 27
_gno. 17
_gp. 4034-4038
856 4 0 _uhttps://doi.org/10.1016/j.bmcl.2017.07.052
_zAvailable from publisher's website
999 _c27432555
_d27432555