000 02075 a2200637 4500
005 20250517150943.0
264 0 _c20171219
008 201712s 0 0 eng d
022 _a1464-3405
024 7 _a10.1016/j.bmcl.2017.04.021
_2doi
040 _aNLM
_beng
_cNLM
100 1 _aHoyt, Scott B
245 0 0 _aDiscovery of indazole aldosterone synthase (CYP11B2) inhibitors as potential treatments for hypertension.
_h[electronic resource]
260 _bBioorganic & medicinal chemistry letters
_c06 2017
300 _a2384-2388 p.
_bdigital
500 _aPublication Type: Journal Article
650 0 4 _aAnimals
650 0 4 _aAntihypertensive Agents
_xchemical synthesis
650 0 4 _aAromatase Inhibitors
_xchemical synthesis
650 0 4 _aCell Line
650 0 4 _aCricetulus
650 0 4 _aCytochrome P-450 CYP11B2
_xantagonists & inhibitors
650 0 4 _aCytochrome P-450 CYP2D6 Inhibitors
_xchemical synthesis
650 0 4 _aHumans
650 0 4 _aHypertension
_xdrug therapy
650 0 4 _aIndazoles
_xchemical synthesis
650 0 4 _aMacaca mulatta
650 0 4 _aMale
650 0 4 _aRats, Sprague-Dawley
650 0 4 _aStereoisomerism
650 0 4 _aSteroid 11-beta-Hydroxylase
_xantagonists & inhibitors
700 1 _aTaylor, Jerry
700 1 _aLondon, Clare
700 1 _aAli, Amjad
700 1 _aUjjainwalla, Feroze
700 1 _aTata, Jim
700 1 _aStruthers, Mary
700 1 _aCully, Doris
700 1 _aWisniewski, Tom
700 1 _aRen, Ning
700 1 _aBopp, Charlene
700 1 _aSok, Andrea
700 1 _aVerras, Andreas
700 1 _aMcMasters, Daniel
700 1 _aChen, Qing
700 1 _aTung, Elaine
700 1 _aTang, Wei
700 1 _aSalituro, Gino
700 1 _aClemas, Joe
700 1 _aZhou, Gaochao
700 1 _aMacNeil, Douglas
700 1 _aDuffy, Ruth
700 1 _aXiong, Yusheng
773 0 _tBioorganic & medicinal chemistry letters
_gvol. 27
_gno. 11
_gp. 2384-2388
856 4 0 _uhttps://doi.org/10.1016/j.bmcl.2017.04.021
_zAvailable from publisher's website
999 _c27087498
_d27087498