000 01926 a2200481 4500
005 20250517132159.0
264 0 _c20181231
008 201812s 0 0 eng d
022 _a2472-5560
024 7 _a10.1177/2472555216679994
_2doi
040 _aNLM
_beng
_cNLM
100 1 _aScharf, Nathan T
245 0 0 _aNovel Chemical Scaffolds for Inhibition of Rifamycin-Resistant RNA Polymerase Discovered from High-Throughput Screening.
_h[electronic resource]
260 _bSLAS discovery : advancing life sciences R & D
_c03 2017
300 _a287-297 p.
_bdigital
500 _aPublication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
650 0 4 _aAntitubercular Agents
_xpharmacology
650 0 4 _aAptamers, Nucleotide
_xgenetics
650 0 4 _aBacterial Proteins
_xantagonists & inhibitors
650 0 4 _aBiological Assay
650 0 4 _aDNA-Directed RNA Polymerases
_xantagonists & inhibitors
650 0 4 _aDrug Discovery
650 0 4 _aDrug Resistance, Bacterial
_xdrug effects
650 0 4 _aEscherichia coli
_xdrug effects
650 0 4 _aExtensively Drug-Resistant Tuberculosis
_xdrug therapy
650 0 4 _aGene Expression
650 0 4 _aHigh-Throughput Screening Assays
650 0 4 _aHumans
650 0 4 _aMicrobial Sensitivity Tests
650 0 4 _aMutation
650 0 4 _aMycobacterium tuberculosis
_xdrug effects
650 0 4 _aPlasmids
_xchemistry
650 0 4 _aRifampin
_xpharmacology
650 0 4 _aRifamycins
_xpharmacology
650 0 4 _aSmall Molecule Libraries
_xchemistry
650 0 4 _aStructure-Activity Relationship
700 1 _aMolodtsov, Vadim
700 1 _aKontos, Arrin
700 1 _aMurakami, Katsuhiko S
700 1 _aGarcia, George A
773 0 _tSLAS discovery : advancing life sciences R & D
_gvol. 22
_gno. 3
_gp. 287-297
856 4 0 _uhttps://doi.org/10.1177/2472555216679994
_zAvailable from publisher's website
999 _c26734982
_d26734982