000 01673 a2200445 4500
005 20250517035520.0
264 0 _c20150914
008 201509s 0 0 eng d
022 _a1520-4804
024 7 _a10.1021/acs.jmedchem.5b00613
_2doi
040 _aNLM
_beng
_cNLM
100 1 _aRan, Xu
245 0 0 _aStructure-Based Design of γ-Carboline Analogues as Potent and Specific BET Bromodomain Inhibitors.
_h[electronic resource]
260 _bJournal of medicinal chemistry
_cJun 2015
300 _a4927-39 p.
_bdigital
500 _aPublication Type: Journal Article; Research Support, N.I.H., Extramural; Research Support, Non-U.S. Gov't
650 0 4 _aAntineoplastic Agents
_xchemistry
650 0 4 _aCarbolines
_xchemistry
650 0 4 _aCell Cycle Proteins
650 0 4 _aCell Line, Tumor
650 0 4 _aCrystallography, X-Ray
650 0 4 _aHumans
650 0 4 _aLeukemia
_xdrug therapy
650 0 4 _aMolecular Docking Simulation
650 0 4 _aNuclear Proteins
_xantagonists & inhibitors
650 0 4 _aProtein Serine-Threonine Kinases
_xantagonists & inhibitors
650 0 4 _aRNA-Binding Proteins
_xantagonists & inhibitors
650 0 4 _aTranscription Factors
_xantagonists & inhibitors
700 1 _aZhao, Yujun
700 1 _aLiu, Liu
700 1 _aBai, Longchuan
700 1 _aYang, Chao-Yie
700 1 _aZhou, Bing
700 1 _aMeagher, Jennifer L
700 1 _aChinnaswamy, Krishnapriya
700 1 _aStuckey, Jeanne A
700 1 _aWang, Shaomeng
773 0 _tJournal of medicinal chemistry
_gvol. 58
_gno. 12
_gp. 4927-39
856 4 0 _uhttps://doi.org/10.1021/acs.jmedchem.5b00613
_zAvailable from publisher's website
999 _c24987418
_d24987418