000 01504 a2200397 4500
005 20250516223749.0
264 0 _c20150406
008 201504s 0 0 eng d
022 _a1464-3391
024 7 _a10.1016/j.bmc.2014.06.050
_2doi
040 _aNLM
_beng
_cNLM
100 1 _aEdupuganti, Ramakrishna
245 0 0 _aSynthesis and biological evaluation of pyrido[2,3-d]pyrimidine-2,4-dione derivatives as eEF-2K inhibitors.
_h[electronic resource]
260 _bBioorganic & medicinal chemistry
_cSep 2014
300 _a4910-6 p.
_bdigital
500 _aPublication Type: Journal Article; Research Support, N.I.H., Extramural
650 0 4 _aDose-Response Relationship, Drug
650 0 4 _aElongation Factor 2 Kinase
_xantagonists & inhibitors
650 0 4 _aHumans
650 0 4 _aMolecular Structure
650 0 4 _aProtein Kinase Inhibitors
_xchemical synthesis
650 0 4 _aPyridines
_xchemical synthesis
650 0 4 _aPyrimidinones
_xchemical synthesis
650 0 4 _aRecombinant Proteins
_xmetabolism
650 0 4 _aStructure-Activity Relationship
650 0 4 _aTumor Cells, Cultured
700 1 _aWang, Qiantao
700 1 _aTavares, Clint D J
700 1 _aChitjian, Catrina A
700 1 _aBachman, James L
700 1 _aRen, Pengyu
700 1 _aAnslyn, Eric V
700 1 _aDalby, Kevin N
773 0 _tBioorganic & medicinal chemistry
_gvol. 22
_gno. 17
_gp. 4910-6
856 4 0 _uhttps://doi.org/10.1016/j.bmc.2014.06.050
_zAvailable from publisher's website
999 _c24029307
_d24029307