000 01729 a2200433 4500
005 20250516155825.0
264 0 _c20140318
008 201403s 0 0 eng d
022 _a1464-3391
024 7 _a10.1016/j.bmc.2013.05.050
_2doi
040 _aNLM
_beng
_cNLM
100 1 _aMajo, Vattoly J
245 0 0 _aSynthesis and in vivo evaluation of [(18)F]2-(4-(4-(2-(2-fluoroethoxy)phenyl)piperazin-1-yl)butyl)-4-methyl-1,2,4-triazine-3,5(2H,4H)-dione ([(18)F]FECUMI-101) as an imaging probe for 5-HT1A receptor agonist in nonhuman primates.
_h[electronic resource]
260 _bBioorganic & medicinal chemistry
_cSep 2013
300 _a5598-604 p.
_bdigital
500 _aPublication Type: Journal Article; Research Support, N.I.H., Extramural
650 0 4 _aAnimals
650 0 4 _aBlood-Brain Barrier
_xmetabolism
650 0 4 _aBrain
_xdiagnostic imaging
650 0 4 _aFluorine Radioisotopes
_xchemistry
650 0 4 _aPapio
650 0 4 _aPiperazines
_xchemical synthesis
650 0 4 _aPositron-Emission Tomography
650 0 4 _aProtein Binding
650 0 4 _aRadiopharmaceuticals
_xchemical synthesis
650 0 4 _aReceptor, Serotonin, 5-HT1A
_xchemistry
650 0 4 _aSerotonin 5-HT1 Receptor Agonists
_xchemical synthesis
650 0 4 _aTriazines
_xchemical synthesis
700 1 _aMilak, Matthew S
700 1 _aPrabhakaran, Jaya
700 1 _aMali, Pratap
700 1 _aSavenkova, Lyudmila
700 1 _aSimpson, Norman R
700 1 _aMann, J John
700 1 _aParsey, Ramin V
700 1 _aKumar, J S Dileep
773 0 _tBioorganic & medicinal chemistry
_gvol. 21
_gno. 17
_gp. 5598-604
856 4 0 _uhttps://doi.org/10.1016/j.bmc.2013.05.050
_zAvailable from publisher's website
999 _c22881461
_d22881461