| 000 | 02164 a2200601 4500 | ||
|---|---|---|---|
| 005 | 20250516145845.0 | ||
| 264 | 0 | _c20131209 | |
| 008 | 201312s 0 0 eng d | ||
| 022 | _a1464-3405 | ||
| 024 | 7 |
_a10.1016/j.bmcl.2013.04.012 _2doi |
|
| 040 |
_aNLM _beng _cNLM |
||
| 100 | 1 | _aChaturvedula, Prasad V | |
| 245 | 0 | 0 |
_aDiscovery of (R)-N-(3-(7-methyl-1H-indazol-5-yl)-1-(4-(1-methylpiperidin-4-yl)-1-oxopropan-2-yl)-4-(2-oxo-1,2-dihydroquinolin-3-yl)piperidine-1-carboxamide (BMS-742413): a potent human CGRP antagonist with superior safety profile for the treatment of migraine through intranasal delivery. _h[electronic resource] |
| 260 |
_bBioorganic & medicinal chemistry letters _cJun 2013 |
||
| 300 |
_a3157-61 p. _bdigital |
||
| 500 | _aPublication Type: Journal Article | ||
| 650 | 0 | 4 | _aAdministration, Intranasal |
| 650 | 0 | 4 |
_aAmides _xchemistry |
| 650 | 0 | 4 | _aAnimals |
| 650 | 0 | 4 | _aCaco-2 Cells |
| 650 | 0 | 4 | _aCalcitonin Gene-Related Peptide Receptor Antagonists |
| 650 | 0 | 4 | _aCallithrix |
| 650 | 0 | 4 |
_aCoronary Vessels _xdrug effects |
| 650 | 0 | 4 | _aDrug Evaluation, Preclinical |
| 650 | 0 | 4 |
_aFace _xblood supply |
| 650 | 0 | 4 | _aHumans |
| 650 | 0 | 4 |
_aIndazoles _xchemistry |
| 650 | 0 | 4 |
_aMigraine Disorders _xdrug therapy |
| 650 | 0 | 4 |
_aQuinolones _xchemistry |
| 650 | 0 | 4 | _aRabbits |
| 650 | 0 | 4 | _aRats |
| 650 | 0 | 4 |
_aReceptors, Calcitonin Gene-Related Peptide _xmetabolism |
| 650 | 0 | 4 |
_aRespiratory Mucosa _xdrug effects |
| 700 | 1 | _aMercer, Stephen E | |
| 700 | 1 | _aPin, Sokhom S | |
| 700 | 1 | _aThalody, George | |
| 700 | 1 | _aXu, Cen | |
| 700 | 1 | _aConway, Charlie M | |
| 700 | 1 | _aKeavy, Deborah | |
| 700 | 1 | _aSignor, Laura | |
| 700 | 1 | _aCantor, Glenn H | |
| 700 | 1 | _aMathias, Neil | |
| 700 | 1 | _aMoench, Paul | |
| 700 | 1 | _aDenton, Rex | |
| 700 | 1 | _aMacci, Robert | |
| 700 | 1 | _aSchartman, Richard | |
| 700 | 1 | _aWhiterock, Valerie | |
| 700 | 1 | _aDavis, Carl | |
| 700 | 1 | _aMacor, John E | |
| 700 | 1 | _aDubowchik, Gene M | |
| 773 | 0 |
_tBioorganic & medicinal chemistry letters _gvol. 23 _gno. 11 _gp. 3157-61 |
|
| 856 | 4 | 0 |
_uhttps://doi.org/10.1016/j.bmcl.2013.04.012 _zAvailable from publisher's website |
| 999 |
_c22712954 _d22712954 |
||