000 02626 a2200805 4500
005 20250516145441.0
264 0 _c20131126
008 201311s 0 0 eng d
022 _a1521-009X
024 7 _a10.1124/dmd.112.050500
_2doi
040 _aNLM
_beng
_cNLM
100 1 _aBentz, Joe
245 0 0 _aVariability in P-glycoprotein inhibitory potency (IC₅₀) using various in vitro experimental systems: implications for universal digoxin drug-drug interaction risk assessment decision criteria.
_h[electronic resource]
260 _bDrug metabolism and disposition: the biological fate of chemicals
_cJul 2013
300 _a1347-66 p.
_bdigital
500 _aPublication Type: Journal Article; Research Support, N.I.H., Extramural
650 0 4 _aATP Binding Cassette Transporter, Subfamily B, Member 1
_xantagonists & inhibitors
650 0 4 _aAnimals
650 0 4 _aBiological Transport
650 0 4 _aCaco-2 Cells
650 0 4 _aDigoxin
_xpharmacokinetics
650 0 4 _aDogs
650 0 4 _aDrug Interactions
650 0 4 _aHumans
650 0 4 _aInhibitory Concentration 50
650 0 4 _aLLC-PK1 Cells
650 0 4 _aPrincipal Component Analysis
650 0 4 _aRisk Assessment
650 0 4 _aSwine
700 1 _aO'Connor, Michael P
700 1 _aBednarczyk, Dallas
700 1 _aColeman, Joann
700 1 _aLee, Caroline
700 1 _aPalm, Johan
700 1 _aPak, Y Anne
700 1 _aPerloff, Elke S
700 1 _aReyner, Eric
700 1 _aBalimane, Praveen
700 1 _aBrännström, Marie
700 1 _aChu, Xiaoyan
700 1 _aFunk, Christoph
700 1 _aGuo, Ailan
700 1 _aHanna, Imad
700 1 _aHerédi-Szabó, Krisztina
700 1 _aHillgren, Kate
700 1 _aLi, Libin
700 1 _aHollnack-Pusch, Evelyn
700 1 _aJamei, Masoud
700 1 _aLin, Xuena
700 1 _aMason, Andrew K
700 1 _aNeuhoff, Sibylle
700 1 _aPatel, Aarti
700 1 _aPodila, Lalitha
700 1 _aPlise, Emile
700 1 _aRajaraman, Ganesh
700 1 _aSalphati, Laurent
700 1 _aSands, Eric
700 1 _aTaub, Mitchell E
700 1 _aTaur, Jan-Shiang
700 1 _aWeitz, Dietmar
700 1 _aWortelboer, Heleen M
700 1 _aXia, Cindy Q
700 1 _aXiao, Guangqing
700 1 _aYabut, Jocelyn
700 1 _aYamagata, Tetsuo
700 1 _aZhang, Lei
700 1 _aEllens, Harma
773 0 _tDrug metabolism and disposition: the biological fate of chemicals
_gvol. 41
_gno. 7
_gp. 1347-66
856 4 0 _uhttps://doi.org/10.1124/dmd.112.050500
_zAvailable from publisher's website
999 _c22702328
_d22702328