000 01484 a2200385 4500
005 20250516115955.0
264 0 _c20130423
008 201304s 0 0 eng d
022 _a1464-3405
024 7 _a10.1016/j.bmcl.2012.09.043
_2doi
040 _aNLM
_beng
_cNLM
100 1 _aZhang, Peng
245 0 0 _aIdentification of novel scaffold of benzothiazepinones as non-ATP competitive glycogen synthase kinase-3β inhibitors through virtual screening.
_h[electronic resource]
260 _bBioorganic & medicinal chemistry letters
_cDec 2012
300 _a7232-6 p.
_bdigital
500 _aPublication Type: Journal Article; Research Support, Non-U.S. Gov't
650 0 4 _aAdenosine Triphosphate
_xmetabolism
650 0 4 _aBinding Sites
650 0 4 _aBinding, Competitive
650 0 4 _aGlycogen Synthase Kinase 3
_xantagonists & inhibitors
650 0 4 _aGlycogen Synthase Kinase 3 beta
650 0 4 _aKinetics
650 0 4 _aMolecular Docking Simulation
650 0 4 _aProtein Binding
650 0 4 _aProtein Kinase Inhibitors
_xchemical synthesis
650 0 4 _aProtein Structure, Tertiary
650 0 4 _aThiazepines
_xchemical synthesis
700 1 _aHu, Hai-Rong
700 1 _aHuang, Zhao-Hui
700 1 _aLei, Jia-Yi
700 1 _aChu, Yong
700 1 _aYe, De-Yong
773 0 _tBioorganic & medicinal chemistry letters
_gvol. 22
_gno. 23
_gp. 7232-6
856 4 0 _uhttps://doi.org/10.1016/j.bmcl.2012.09.043
_zAvailable from publisher's website
999 _c22213623
_d22213623