000 | 01771 a2200541 4500 | ||
---|---|---|---|
005 | 20250516114151.0 | ||
264 | 0 | _c20130429 | |
008 | 201304s 0 0 eng d | ||
022 | _a1860-7187 | ||
024 | 7 |
_a10.1002/cmdc.201200406 _2doi |
|
040 |
_aNLM _beng _cNLM |
||
100 | 1 | _aProvins, Laurent | |
245 | 0 | 0 |
_aLead optimization of thiazolo[5,4-c]piperidines: 3-cyclobutoxy linker as a key spacer for H(3)R inverse agonists. _h[electronic resource] |
260 |
_bChemMedChem _cDec 2012 |
||
300 |
_a2087-92 p. _bdigital |
||
500 | _aPublication Type: Journal Article; Research Support, Non-U.S. Gov't | ||
650 | 0 | 4 | _aAnimals |
650 | 0 | 4 |
_aBenzamides _xchemistry |
650 | 0 | 4 | _aCaco-2 Cells |
650 | 0 | 4 |
_aHistamine Agonists _xchemistry |
650 | 0 | 4 | _aHumans |
650 | 0 | 4 | _aMale |
650 | 0 | 4 |
_aPiperidines _xchemistry |
650 | 0 | 4 | _aRats |
650 | 0 | 4 | _aRats, Wistar |
650 | 0 | 4 |
_aReceptors, Histamine H3 _xmetabolism |
650 | 0 | 4 | _aStructure-Activity Relationship |
650 | 0 | 4 |
_aThiazoles _xchemistry |
650 | 0 | 4 |
_aTrans-Activators _xmetabolism |
650 | 0 | 4 | _aTranscriptional Regulator ERG |
700 | 1 | _aDenonne, Frédéric | |
700 | 1 | _aCélanire, Sylvain | |
700 | 1 | _aChristophe, Bernard | |
700 | 1 | _aDefays, Sabine | |
700 | 1 | _aDelaunoy, Christel | |
700 | 1 | _aDelporte, Marie-Laure | |
700 | 1 | _aDemaude, Thierry | |
700 | 1 | _aDurieu, Véronique | |
700 | 1 | _aGillard, Michel | |
700 | 1 | _aHubert, Delphine | |
700 | 1 | _aLamberty, Yves | |
700 | 1 | _aLorent, Geneviève | |
700 | 1 | _aValade, Anne | |
700 | 1 | _aVanbellinghen, Alain | |
700 | 1 | _aVan Houtvin, Nathalie | |
773 | 0 |
_tChemMedChem _gvol. 7 _gno. 12 _gp. 2087-92 |
|
856 | 4 | 0 |
_uhttps://doi.org/10.1002/cmdc.201200406 _zAvailable from publisher's website |
999 |
_c22164281 _d22164281 |