000 02068 a2200541 4500
005 20250516074407.0
264 0 _c20120525
008 201205s 0 0 eng d
022 _a1520-4804
024 7 _a10.1021/jm201438f
_2doi
040 _aNLM
_beng
_cNLM
100 1 _aCaboni, Laura
245 0 0 _a"True" antiandrogens-selective non-ligand-binding pocket disruptors of androgen receptor-coactivator interactions: novel tools for prostate cancer.
_h[electronic resource]
260 _bJournal of medicinal chemistry
_cFeb 2012
300 _a1635-44 p.
_bdigital
500 _aPublication Type: Journal Article; Research Support, Non-U.S. Gov't
650 0 4 _aAndrogen Antagonists
_xchemical synthesis
650 0 4 _aAntineoplastic Agents
_xchemical synthesis
650 0 4 _aCell Proliferation
_xdrug effects
650 0 4 _aCell Survival
_xdrug effects
650 0 4 _aDatabases, Factual
650 0 4 _aDrug Screening Assays, Antitumor
650 0 4 _aEstrogen Receptor alpha
_xmetabolism
650 0 4 _aEstrogen Receptor beta
_xmetabolism
650 0 4 _aFluorescence Polarization
650 0 4 _aFluorescence Resonance Energy Transfer
650 0 4 _aHumans
650 0 4 _aHydrazines
_xchemical synthesis
650 0 4 _aMale
650 0 4 _aModels, Molecular
650 0 4 _aNuclear Receptor Coactivators
_xmetabolism
650 0 4 _aProstate-Specific Antigen
_xmetabolism
650 0 4 _aProstatic Neoplasms
_xdrug therapy
650 0 4 _aReceptors, Androgen
_xmetabolism
650 0 4 _aReceptors, Glucocorticoid
_xmetabolism
650 0 4 _aReceptors, Progesterone
_xantagonists & inhibitors
650 0 4 _aStructure-Activity Relationship
700 1 _aKinsella, Gemma K
700 1 _aBlanco, Fernando
700 1 _aFayne, Darren
700 1 _aJagoe, William N
700 1 _aCarr, Miriam
700 1 _aWilliams, D Clive
700 1 _aMeegan, Mary J
700 1 _aLloyd, David G
773 0 _tJournal of medicinal chemistry
_gvol. 55
_gno. 4
_gp. 1635-44
856 4 0 _uhttps://doi.org/10.1021/jm201438f
_zAvailable from publisher's website
999 _c21494213
_d21494213