000 01307 a2200325 4500
005 20250516060501.0
264 0 _c20120213
008 201202s 0 0 eng d
022 _a1464-3405
024 7 _a10.1016/j.bmcl.2011.09.044
_2doi
040 _aNLM
_beng
_cNLM
100 1 _aMatthews, Hayden
245 0 0 _aSynthesis and preliminary evaluation of amiloride analogs as inhibitors of the urokinase-type plasminogen activator (uPA).
_h[electronic resource]
260 _bBioorganic & medicinal chemistry letters
_cNov 2011
300 _a6760-6 p.
_bdigital
500 _aPublication Type: Journal Article; Research Support, Non-U.S. Gov't
650 0 4 _aAmiloride
_xanalogs & derivatives
650 0 4 _aAntineoplastic Agents
_xchemical synthesis
650 0 4 _aDiuretics
_xchemical synthesis
650 0 4 _aHumans
650 0 4 _aModels, Molecular
650 0 4 _aNeoplasms
_xdrug therapy
650 0 4 _aStructure-Activity Relationship
650 0 4 _aUrokinase-Type Plasminogen Activator
_xantagonists & inhibitors
700 1 _aRanson, Marie
700 1 _aTyndall, Joel D A
700 1 _aKelso, Michael J
773 0 _tBioorganic & medicinal chemistry letters
_gvol. 21
_gno. 22
_gp. 6760-6
856 4 0 _uhttps://doi.org/10.1016/j.bmcl.2011.09.044
_zAvailable from publisher's website
999 _c21213252
_d21213252