000 01571 a2200445 4500
005 20250516055614.0
264 0 _c20120207
008 201202s 0 0 eng d
022 _a1520-4804
024 7 _a10.1021/jm200981s
_2doi
040 _aNLM
_beng
_cNLM
100 1 _aVidal-Mosquera, Miquel
245 0 0 _aTriazine-based vanilloid 1 receptor open channel blockers: design, synthesis, evaluation, and SAR analysis.
_h[electronic resource]
260 _bJournal of medicinal chemistry
_cNov 2011
300 _a7441-52 p.
_bdigital
500 _aPublication Type: Journal Article; Research Support, Non-U.S. Gov't
650 0 4 _aAnalgesics
_xchemical synthesis
650 0 4 _aAnimals
650 0 4 _aBinding Sites
650 0 4 _aDrug Design
650 0 4 _aFemale
650 0 4 _aOocytes
_xdrug effects
650 0 4 _aPatch-Clamp Techniques
650 0 4 _aRats
650 0 4 _aRecombinant Proteins
_xantagonists & inhibitors
650 0 4 _aStructure-Activity Relationship
650 0 4 _aTRPV Cation Channels
_xantagonists & inhibitors
650 0 4 _aTriazines
_xchemical synthesis
650 0 4 _aXenopus
700 1 _aFernández-Carvajal, Asia
700 1 _aMoure, Alejandra
700 1 _aValente, Pierluigi
700 1 _aPlanells-Cases, Rosa
700 1 _aGonzález-Ros, José M
700 1 _aBujons, Jordi
700 1 _aFerrer-Montiel, Antonio
700 1 _aMesseguer, Angel
773 0 _tJournal of medicinal chemistry
_gvol. 54
_gno. 21
_gp. 7441-52
856 4 0 _uhttps://doi.org/10.1021/jm200981s
_zAvailable from publisher's website
999 _c21187942
_d21187942