000 01509 a2200433 4500
005 20250516030222.0
264 0 _c20110721
008 201107s 0 0 eng d
022 _a1860-7187
024 7 _a10.1002/cmdc.201100047
_2doi
040 _aNLM
_beng
_cNLM
100 1 _aKeil, Stefanie
245 0 0 _aSulfonylthiadiazoles with an unusual binding mode as partial dual peroxisome proliferator-activated receptor (PPAR) γ/δ agonists with high potency and in vivo efficacy.
_h[electronic resource]
260 _bChemMedChem
_cApr 2011
300 _a633-53 p.
_bdigital
500 _aPublication Type: Journal Article
650 0 4 _aAnimals
650 0 4 _aBinding Sites
650 0 4 _aCrystallography, X-Ray
650 0 4 _aDiabetes Mellitus, Experimental
_xdrug therapy
650 0 4 _aDiabetes Mellitus, Type 2
_xdrug therapy
650 0 4 _aMice
650 0 4 _aPPAR delta
_xagonists
650 0 4 _aPPAR gamma
_xagonists
650 0 4 _aStructure-Activity Relationship
650 0 4 _aSulfones
_xagonists
650 0 4 _aThiadiazoles
_xagonists
700 1 _aMatter, Hans
700 1 _aSchönafinger, Karl
700 1 _aGlien, Maike
700 1 _aMathieu, Magali
700 1 _aMarquette, Jean-Pierre
700 1 _aMichot, Nadine
700 1 _aHaag-Diergarten, Silke
700 1 _aUrmann, Matthias
700 1 _aWendler, Wolfgang
773 0 _tChemMedChem
_gvol. 6
_gno. 4
_gp. 633-53
856 4 0 _uhttps://doi.org/10.1002/cmdc.201100047
_zAvailable from publisher's website
999 _c20672032
_d20672032