000 | 01422 a2200421 4500 | ||
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005 | 20250516023707.0 | ||
264 | 0 | _c20110705 | |
008 | 201107s 0 0 eng d | ||
022 | _a1464-3405 | ||
024 | 7 |
_a10.1016/j.bmcl.2011.01.093 _2doi |
|
040 |
_aNLM _beng _cNLM |
||
100 | 1 | _aHudson, Andrew R | |
245 | 0 | 0 |
_aDiscovery of orally available tetrahydroquinoline-based glucocorticoid receptor agonists. _h[electronic resource] |
260 |
_bBioorganic & medicinal chemistry letters _cMar 2011 |
||
300 |
_a1697-700 p. _bdigital |
||
500 | _aPublication Type: Journal Article | ||
650 | 0 | 4 | _aAdministration, Oral |
650 | 0 | 4 | _aAnimals |
650 | 0 | 4 | _aDrug Discovery |
650 | 0 | 4 | _aEnzyme-Linked Immunosorbent Assay |
650 | 0 | 4 | _aHumans |
650 | 0 | 4 |
_aQuinolines _xadministration & dosage |
650 | 0 | 4 | _aRats |
650 | 0 | 4 | _aRats, Sprague-Dawley |
650 | 0 | 4 |
_aReceptors, Glucocorticoid _xagonists |
650 | 0 | 4 | _aStructure-Activity Relationship |
700 | 1 | _aHiguchi, Robert I | |
700 | 1 | _aRoach, Steven L | |
700 | 1 | _aAdams, Mark E | |
700 | 1 | _aVassar, Angela | |
700 | 1 | _aSyka, Peter M | |
700 | 1 | _aMais, Dale E | |
700 | 1 | _aMiner, Jeffrey N | |
700 | 1 | _aMarschke, Keith B | |
700 | 1 | _aZhi, Lin | |
773 | 0 |
_tBioorganic & medicinal chemistry letters _gvol. 21 _gno. 6 _gp. 1697-700 |
|
856 | 4 | 0 |
_uhttps://doi.org/10.1016/j.bmcl.2011.01.093 _zAvailable from publisher's website |
999 |
_c20594427 _d20594427 |