000 01546 a2200433 4500
005 20250515195805.0
264 0 _c20100420
008 201004s 0 0 eng d
022 _a1464-3405
024 7 _a10.1016/j.bmcl.2009.11.078
_2doi
040 _aNLM
_beng
_cNLM
100 1 _aSabbatini, Fabio M
245 0 0 _aSynthesis and pharmacological characterization of constrained analogues of Vestipitant as in vitro potent and orally active NK(1) receptor antagonists.
_h[electronic resource]
260 _bBioorganic & medicinal chemistry letters
_cJan 2010
300 _a623-7 p.
_bdigital
500 _aPublication Type: Journal Article
650 0 4 _aAnti-Anxiety Agents
_xchemical synthesis
650 0 4 _aDrug Design
650 0 4 _aFluorobenzenes
650 0 4 _aHumans
650 0 4 _aMolecular Conformation
650 0 4 _aNeurokinin-1 Receptor Antagonists
650 0 4 _aPiperidines
_xchemical synthesis
650 0 4 _aReceptors, Neurokinin-1
_xmetabolism
700 1 _aDi Fabio, Romano
700 1 _aGriffante, Cristiana
700 1 _aPentassuglia, Giorgio
700 1 _aZonzini, Laura
700 1 _aMelotto, Sergio
700 1 _aAlvaro, Giuseppe
700 1 _aCapelli, Anna M
700 1 _aPippo, Lara
700 1 _aPerdona', Elisabetta
700 1 _aSt Denis, Yves
700 1 _aCosta, Silvano
700 1 _aCorsi, Mauro
773 0 _tBioorganic & medicinal chemistry letters
_gvol. 20
_gno. 2
_gp. 623-7
856 4 0 _uhttps://doi.org/10.1016/j.bmcl.2009.11.078
_zAvailable from publisher's website
999 _c19346166
_d19346166