000 01486 a2200433 4500
005 20250515183124.0
264 0 _c20091123
008 200911s 0 0 eng d
022 _a1464-3405
024 7 _a10.1016/j.bmcl.2009.07.109
_2doi
040 _aNLM
_beng
_cNLM
100 1 _aSubrath, Joan
245 0 0 _aC-5 Substituted heteroaryl 3-pyridinecarbonitriles as PKCtheta inhibitors: Part I.
_h[electronic resource]
260 _bBioorganic & medicinal chemistry letters
_cSep 2009
300 _a5423-5 p.
_bdigital
500 _aPublication Type: Journal Article
650 0 4 _aAnimals
650 0 4 _aInhibitory Concentration 50
650 0 4 _aIsoenzymes
_xantagonists & inhibitors
650 0 4 _aMice
650 0 4 _aMice, Knockout
650 0 4 _aNitriles
_xchemistry
650 0 4 _aProtein Kinase C
_xantagonists & inhibitors
650 0 4 _aProtein Kinase C-theta
650 0 4 _aProtein Kinase Inhibitors
_xchemistry
650 0 4 _aPyridines
_xchemistry
650 0 4 _aStructure-Activity Relationship
650 0 4 _aT-Lymphocytes
_xdrug effects
700 1 _aWang, Daniel
700 1 _aWu, Biqi
700 1 _aNiu, Chuansheng
700 1 _aBoschelli, Diane H
700 1 _aLee, Julie
700 1 _aYang, Xiaoke
700 1 _aBrennan, Agnes
700 1 _aChaudhary, Divya
773 0 _tBioorganic & medicinal chemistry letters
_gvol. 19
_gno. 18
_gp. 5423-5
856 4 0 _uhttps://doi.org/10.1016/j.bmcl.2009.07.109
_zAvailable from publisher's website
999 _c19086212
_d19086212