000			02063 a2200589 4500
005			20250515095008.0
264		0	_c20080403
008			200804s 0 0 eng d
022			_a0022-2623
024	7		_a10.1021/jm070778w _2doi
040			_aNLM _beng _cNLM
100	1		_aBiggadike, Keith
245	0	0	_aNonsteroidal glucocorticoid agonists: tetrahydronaphthalenes with alternative steroidal A-ring mimetics possessing dissociated (transrepression/transactivation) efficacy selectivity. _h[electronic resource]
260			_bJournal of medicinal chemistry _cDec 2007
300			_a6519-34 p. _bdigital
500			_aPublication Type: Journal Article
650	0	4	_aAnti-Inflammatory Agents, Non-Steroidal _xchemical synthesis
650	0	4	_aBinding Sites
650	0	4	_aCell Line
650	0	4	_aDrug Partial Agonism
650	0	4	_aHumans
650	0	4	_aMammary Tumor Virus, Mouse _xgenetics
650	0	4	_aModels, Molecular
650	0	4	_aMolecular Mimicry
650	0	4	_aNF-kappa B _xgenetics
650	0	4	_aReceptors, Glucocorticoid _xagonists
650	0	4	_aStereoisomerism
650	0	4	_aStructure-Activity Relationship
650	0	4	_aTetrahydronaphthalenes _xchemical synthesis
650	0	4	_aTranscription, Genetic _xdrug effects
650	0	4	_aTranscriptional Activation _xdrug effects
700	1		_aBoudjelal, Mohamed
700	1		_aClackers, Margaret
700	1		_aCoe, Diane M
700	1		_aDemaine, Derek A
700	1		_aHardy, George W
700	1		_aHumphreys, Davina
700	1		_aInglis, Graham G A
700	1		_aJohnston, Michael J
700	1		_aJones, Haydn T
700	1		_aHouse, David
700	1		_aLoiseau, Richard
700	1		_aNeedham, Deborah
700	1		_aSkone, Philip A
700	1		_aUings, Iain
700	1		_aVeitch, Gemma
700	1		_aWeingarten, Gordon G
700	1		_aMcLay, Iain M
700	1		_aMacdonald, Simon J F
773	0		_tJournal of medicinal chemistry _gvol. 50 _gno. 26 _gp. 6519-34
856	4	0	_uhttps://doi.org/10.1021/jm070778w _zAvailable from publisher's website
999			_c17554223 _d17554223