000 02043 a2200601 4500
005 20250515093747.0
264 0 _c20080723
008 200807s 0 0 eng d
022 _a1860-7187
024 7 _a10.1002/cmdc.200700230
_2doi
040 _aNLM
_beng
_cNLM
100 1 _aSabbatini, Fabio Maria
245 0 0 _aHeteroaryl-substituted 4-(1H-pyrazol-1-yl)-5,6-dihydro-1H-pyrrolo[2,3-d]pyrimidine derivatives as potent and selective corticotropin-releasing factor receptor-1 antagonists.
_h[electronic resource]
260 _bChemMedChem
_cFeb 2008
300 _a226-9 p.
_bdigital
500 _aPublication Type: Journal Article
650 0 4 _aAnimals
650 0 4 _aAnxiety
_xdrug therapy
650 0 4 _aCorticotropin-Releasing Hormone
_xmetabolism
650 0 4 _aDepression
_xdrug therapy
650 0 4 _aDrug Design
650 0 4 _aModels, Chemical
650 0 4 _aPyrazoles
_xchemical synthesis
650 0 4 _aPyrimidines
_xchemical synthesis
650 0 4 _aRats
650 0 4 _aRats, Wistar
650 0 4 _aReceptors, Corticotropin-Releasing Hormone
_xantagonists & inhibitors
650 0 4 _aStructure-Activity Relationship
650 0 4 _aCRF Receptor, Type 1
700 1 _aDi Fabio, Romano
700 1 _aSt-Denis, Yves
700 1 _aCapelli, Anna-Maria
700 1 _aCastiglioni, Emiliano
700 1 _aContini, Stefania
700 1 _aDonati, Daniele
700 1 _aFazzolari, Elettra
700 1 _aGentile, Gabriella
700 1 _aMicheli, Fabrizio
700 1 _aPavone, Francesca
700 1 _aRinaldi, Marilisa
700 1 _aPasquarello, Alessandra
700 1 _aZampori, Maria Grazia
700 1 _aDi Felice, Pina
700 1 _aZarantonello, Paola
700 1 _aArban, Roberto
700 1 _aPerini, Benedetta
700 1 _aVitulli, Giovanni
700 1 _aBenedetti, Roberto
700 1 _aOliosi, Beatrice
700 1 _aWorby, Angela
773 0 _tChemMedChem
_gvol. 3
_gno. 2
_gp. 226-9
856 4 0 _uhttps://doi.org/10.1002/cmdc.200700230
_zAvailable from publisher's website
999 _c17518063
_d17518063