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3-Substituted Quinolines as RORγt Inverse Agonists. [electronic resource] by
- Tanis, Virginia M
- Venkatesan, Hariharan
- Cummings, Maxwell D
- Albers, Michael
- Kent Barbay, J
- Herman, Krystal
- Kummer, David A
- Milligan, Cynthia
- Nelen, Marina I
- Nishimura, Rachel
- Schlueter, Thomas
- Scott, Brian
- Spurlino, John
- Wolin, Ronald
- Woods, Craig
- Xue, Xiaohua
- Edwards, James P
- Fourie, Anne M
- Leonard, Kristi
Producer: 20200921
In:
Bioorganic & medicinal chemistry letters vol. 29
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Tetrahydroindazole derivatives as potent and peripherally selective cannabinoid-1 (CB1) receptor inverse agonists. [electronic resource] by
- Matthews, Jay M
- McNally, James J
- Connolly, Peter J
- Xia, Mingde
- Zhu, Bin
- Black, Shawn
- Chen, Cailin
- Hou, Cuifen
- Liang, Yin
- Tang, Yuting
- Macielag, Mark J
Producer: 20170717
In:
Bioorganic & medicinal chemistry letters vol. 26
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Hemopressin is an inverse agonist of CB1 cannabinoid receptors. [electronic resource] by
- Heimann, Andrea S
- Gomes, Ivone
- Dale, Camila S
- Pagano, Rosana L
- Gupta, Achla
- de Souza, Laura L
- Luchessi, Augusto D
- Castro, Leandro M
- Giorgi, Renata
- Rioli, Vanessa
- Ferro, Emer S
- Devi, Lakshmi A
Producer: 20080128
In:
Proceedings of the National Academy of Sciences of the United States of America vol. 104
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Metabolism and excretion of [14C]taranabant, a cannabinoid-1 inverse agonist, in humans. [electronic resource] by
- Karanam, Bindhu
- Addy, Carol
- Bateman, Thomas
- Reddy, Vijay Bhasker
- Li, Susie
- Dean, Dennis
- Li, Hankun
- Jones, Allen
- Schenk, David
- Zhang, Andy Shiqiang
- Braun, Matt
- Freeman, Amanda
- Flach, Stephen
- Stoch, Aubrey
- Chodakewitz, Jeff
- Wagner, John A
- Kumar, Sanjeev
Producer: 20110104
In:
Xenobiotica; the fate of foreign compounds in biological systems vol. 40
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Discovery of oxa-sultams as RORc inverse agonists showing reduced lipophilicity, improved selectivity and favorable ADME properties. [electronic resource] by
- René, Olivier
- Fauber, Benjamin P
- Barnard, Adrian
- Chapman, Kerry
- Deng, Yuzhong
- Eidenschenk, Céline
- Everett, Christine
- Gobbi, Alberto
- Johnson, Adam R
- La, Hank
- Norman, Maxine
- Salmon, Gary
- Summerhill, Susan
- Wong, Harvey
Producer: 20170808
In:
Bioorganic & medicinal chemistry letters vol. 26
Availability: No items available.
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