N'-(arylsulfonyl)pyrazoline-1-carboxamidines as novel, neutral 5-hydroxytryptamine 6 receptor (5-HT₆R) antagonists with unique structural features. [electronic resource]
Producer: 20120103Description: 7030-54 p. digitalISSN:- 1520-4804
- Amidines -- chemical synthesis
- Animals
- CHO Cells
- Cricetinae
- Cricetulus
- Crystallography, X-Ray
- Guinea Pigs
- Hepatocytes -- metabolism
- Humans
- In Vitro Techniques
- Ligands
- Magnetic Resonance Spectroscopy
- Male
- Models, Molecular
- Protein Binding
- Pyrazoles -- chemical synthesis
- Rats
- Rats, Wistar
- Receptors, Serotonin -- metabolism
- Serotonin Antagonists -- chemical synthesis
- Stereoisomerism
- Structure-Activity Relationship
- Sulfonamides -- chemical synthesis
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Publication Type: Journal Article
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