Results
|
1.
|
|
|
2.
|
Stable pantothenamide bioisosteres: novel antibiotics for Gram-positive bacteria. [electronic resource] by
- Jansen, Patrick A M
- van der Krieken, Danique A
- Botman, Peter N M
- Blaauw, Richard H
- Cavina, Lorenzo
- Raaijmakers, Eline M
- de Heuvel, Erik
- Sandrock, Julia
- Pennings, Lian J
- Hermkens, Pedro H H
- Zeeuwen, Patrick L J M
- Rutjes, Floris P J T
- Schalkwijk, Joost
Producer: 20200225
In:
The Journal of antibiotics vol. 72
Availability: No items available.
|
|
3.
|
Discovery of small molecule vanin inhibitors: new tools to study metabolism and disease. [electronic resource] by
- Jansen, Patrick A M
- van Diepen, Janna A
- Ritzen, Bas
- Zeeuwen, Patrick L J M
- Cacciatore, Ivana
- Cornacchia, Catia
- van Vlijmen-Willems, Ivonne M J J
- de Heuvel, Erik
- Botman, Peter N M
- Blaauw, Richard H
- Hermkens, Pedro H H
- Rutjes, Floris P J T
- Schalkwijk, Joost
Producer: 20141224
In:
ACS chemical biology vol. 8
Availability: No items available.
|
|
4.
|
Alkynamide phthalazinones as a new class of TbrPDEB1 inhibitors (Part 2). [electronic resource] by
- de Heuvel, Erik
- Singh, Abhimanyu K
- Boronat, Pierre
- Kooistra, Albert J
- van der Meer, Tiffany
- Sadek, Payman
- Blaazer, Antoni R
- Shaner, Nathan C
- Bindels, Daphne S
- Caljon, Guy
- Maes, Louis
- Sterk, Geert Jan
- Siderius, Marco
- Oberholzer, Michael
- de Esch, Iwan J P
- Brown, David G
- Leurs, Rob
Producer: 20200917
In:
Bioorganic & medicinal chemistry vol. 27
Availability: No items available.
|
|
5.
|
Evaluation of phthalazinone phosphodiesterase inhibitors with improved activity and selectivity against Trypanosoma cruzi. [electronic resource] by
- De Araújo, Julianna Siciliano
- da Silva, Patrícia Bernardino
- Batista, Marcos Meuser
- Peres, Raiza Brandão
- Cardoso-Santos, Camila
- Kalejaiye, Titilola D
- Munday, Jane C
- De Heuvel, Erik
- Sterk, Geert Jan
- Augustyns, Koen
- Salado, Irene G
- Matheeussen, An
- De Esch, Iwan
- De Koning, Harry P
- Leurs, Rob
- Maes, Louis
- Soeiro, Maria de Nazaré Correia
Producer: 20210624
In:
The Journal of antimicrobial chemotherapy vol. 75
Availability: No items available.
|
|
6.
|
Alkynamide phthalazinones as a new class of TbrPDEB1 inhibitors. [electronic resource] by
- de Heuvel, Erik
- Singh, Abhimanyu K
- Edink, Ewald
- van der Meer, Tiffany
- van der Woude, Melanie
- Sadek, Payman
- Krell-Jørgensen, Mikkel P
- van den Bergh, Toine
- Veerman, Johan
- Caljon, Guy
- Kalejaiye, Titilola D
- Wijtmans, Maikel
- Maes, Louis
- de Koning, Harry P
- Jan Sterk, Geert
- Siderius, Marco
- de Esch, Iwan J P
- Brown, David G
- Leurs, Rob
Producer: 20200917
In:
Bioorganic & medicinal chemistry vol. 27
Availability: No items available.
|
|
7.
|
Screening of a PDE-focused library identifies imidazoles with in vitro and in vivo antischistosomal activity. [electronic resource] by
- Botros, Sanaa S
- William, Samia
- Sabra, Abdel-Nasser A
- El-Lakkany, Naglaa M
- Seif El-Din, Sayed H
- García-Rubia, Alfonso
- Sebastián-Pérez, Victor
- Blaazer, Antoni R
- de Heuvel, Erik
- Sijm, Maarten
- Zheng, Yang
- Salado, Irene G
- Munday, Jane C
- Maes, Louis
- de Esch, Iwan J P
- Sterk, Geert J
- Augustyns, Koen
- Leurs, Rob
- Gil, Carmen
- De Koning, Harry P
Producer: 20191121
In:
International journal for parasitology. Drugs and drug resistance vol. 9
Availability: No items available.
|
|
8.
|
Targeting a Subpocket in Trypanosoma brucei Phosphodiesterase B1 (TbrPDEB1) Enables the Structure-Based Discovery of Selective Inhibitors with Trypanocidal Activity. [electronic resource] by
- Blaazer, Antoni R
- Singh, Abhimanyu K
- de Heuvel, Erik
- Edink, Ewald
- Orrling, Kristina M
- Veerman, Johan J N
- van den Bergh, Toine
- Jansen, Chimed
- Balasubramaniam, Erin
- Mooij, Wouter J
- Custers, Hans
- Sijm, Maarten
- Tagoe, Daniel N A
- Kalejaiye, Titilola D
- Munday, Jane C
- Tenor, Hermann
- Matheeussen, An
- Wijtmans, Maikel
- Siderius, Marco
- de Graaf, Chris
- Maes, Louis
- de Koning, Harry P
- Bailey, David S
- Sterk, Geert Jan
- de Esch, Iwan J P
- Brown, David G
- Leurs, Rob
Producer: 20190528
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
|