Improvement of cyclophosphamide activation by CYP2B6 mutants: from in silico to ex vivo. [electronic resource]
Producer: 20080403Description: 1122-33 p. digitalISSN:- 1521-0111
- Amino Acid Sequence
- Antineoplastic Agents, Alkylating -- metabolism
- Aryl Hydrocarbon Hydroxylases -- chemistry
- Binding Sites
- Cell Death -- drug effects
- Cell Line, Tumor
- Computational Biology -- methods
- Cyclophosphamide -- metabolism
- Cytochrome P-450 CYP2B6
- Humans
- Hydroxylation -- drug effects
- Kinetics
- Ligands
- Microsomes -- drug effects
- Mixed Function Oxygenases -- metabolism
- Models, Molecular
- Molecular Sequence Data
- Mutagenesis
- Mutant Proteins -- metabolism
- Oxidoreductases, N-Demethylating -- chemistry
- Prodrugs -- metabolism
- Saccharomyces cerevisiae -- enzymology
- Sequence Alignment
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Publication Type: Journal Article; Research Support, Non-U.S. Gov't
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