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Prediction of in vivo enantiomeric compositions by modeling in vitro metabolic profiles. [electronic resource] by
- Wang, Mengmeng
- Wang, Qi
- Cai, Hong
- Sleczka, Bogdan
- D'Arienzo, Celia
- Josephs, Jonathan
- Ye, Xiang-Yang
- Robl, Jeffrey
- Gordon, David
- Rodrigues, David
- Harper, Timothy
Producer: 20100802
In:
Journal of pharmaceutical sciences vol. 99
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Synthesis and structure-activity relationship of dihydrobenzofuran derivatives as novel human GPR119 agonists. [electronic resource] by
- Ye, Xiang-Yang
- Morales, Christian L
- Wang, Ying
- Rossi, Karen A
- Malmstrom, Sarah E
- Abousleiman, Mojgan
- Sereda, Larisa
- Apedo, Atsu
- Robl, Jeffrey A
- Miller, Keith J
- Krupinski, John
- Wacker, Dean A
Producer: 20150102
In:
Bioorganic & medicinal chemistry letters vol. 24
Availability: No items available.
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9.
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Design, synthesis, and SAR studies of novel polycyclic acids as potent and selective inhibitors of human 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD-1). [electronic resource] by
- Ye, Xiang-Yang
- Chen, Stephanie Y
- Nayeem, Akbar
- Golla, Rajasree
- Seethala, Ramakrishna
- Wang, Mengmeng
- Harper, Timothy
- Sleczka, Bogdan G
- Li, Yi-Xin
- He, Bin
- Kirby, Mark
- Gordon, David A
- Robl, Jeffrey A
Producer: 20120213
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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10.
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Design, synthesis, and structure-activity relationships of piperidine and dehydropiperidine carboxylic acids as novel, potent dual PPARalpha/gamma agonists. [electronic resource] by
- Ye, Xiang-Yang
- Li, Yi-Xin
- Farrelly, Dennis
- Flynn, Neil
- Gu, Liqun
- Locke, Kenneth T
- Lippy, Jonathan
- O'Malley, Kevin
- Twamley, Celeste
- Zhang, Litao
- Ryono, Denis E
- Zahler, Robert
- Hariharan, Narayanan
- Cheng, Peter T W
Producer: 20080825
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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11.
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Synthesis and structure-activity relationship of 2-adamantylmethyl tetrazoles as potent and selective inhibitors of human 11β-hydroxysteroid dehydrogenase type 1 (11β-HSD1). [electronic resource] by
- Ye, Xiang-Yang
- Yoon, David
- Chen, Stephanie Y
- Nayeem, Akbar
- Golla, Rajasree
- Seethala, Ramakrishna
- Wang, Mengmeng
- Harper, Timothy
- Sleczka, Bogdan G
- Apedo, Atsu
- Li, Yi-Xin
- He, Bin
- Kirby, Mark
- Gordon, David A
- Robl, Jeffrey A
Producer: 20140826
In:
Bioorganic & medicinal chemistry letters vol. 24
Availability: No items available.
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12.
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Synthesis and structure-activity relationships of 2-aryl-4-oxazolylmethoxy benzylglycines and 2-aryl-4-thiazolylmethoxy benzylglycines as novel, potent PPARalpha selective activators- PPARalpha and PPARgamma selectivity modulation. [electronic resource] by
- Ye, Xiang-Yang
- Chen, Stephanie
- Zhang, Hao
- Locke, Kenneth T
- O'Malley, Kevin
- Zhang, Litao
- Srivastava, Raijit
- Miao, Bowman
- Meyers, Daniel
- Monshizadegan, Hossain
- Search, Debra
- Grimm, Denise
- Zhang, Rongan
- Lippy, Jonathan
- Twamley, Celeste
- Muckelbauer, Jodi K
- Chang, Chiehying
- An, Yongmi
- Hosagrahara, Vinayak
- Zhang, Lisa
- Yang, T-J
- Mukherjee, Ranjan
- Cheng, Peter T W
- Tino, Joseph A
Producer: 20100727
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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13.
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Utilization of an Active Site Mutant Receptor for the Identification of Potent and Selective Atypical 5-HT [electronic resource] by
- Carpenter, Joseph
- Wang, Ying
- Wu, Gang
- Feng, Jianxin
- Ye, Xiang-Yang
- Morales, Christian L
- Broekema, Matthias
- Rossi, Karen A
- Miller, Keith J
- Murphy, Brian J
- Wu, Ginger
- Malmstrom, Sarah E
- Azzara, Anthony V
- Sher, Philip M
- Fevig, John M
- Alt, Andrew
- Bertekap, Robert L
- Cullen, Mary Jane
- Harper, Timothy M
- Foster, Kimberly
- Luk, Emily
- Xiang, Qian
- Grubb, Mary F
- Robl, Jeffrey A
- Wacker, Dean A
Producer: 20170905
In:
Journal of medicinal chemistry vol. 60
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14.
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Discovery of Clinical Candidate BMS-823778 as an Inhibitor of Human 11β-Hydroxysteroid Dehydrogenase Type 1 (11β-HSD-1). [electronic resource] by
- Li, Jun
- Kennedy, Lawrence J
- Walker, Steven J
- Wang, Haixia
- Li, James J
- Hong, Zhenqiu
- O'Connor, Stephen P
- Ye, Xiang-Yang
- Chen, Stephanie
- Wu, Shung
- Yoon, David S
- Nayeem, Akbar
- Camac, Daniel M
- Ramamurthy, Vidhyashankar
- Morin, Paul E
- Sheriff, Steven
- Wang, Mengmeng
- Harper, Timothy W
- Golla, Rajasree
- Seethala, Ramakrishna
- Harrity, Thomas
- Ponticiello, Randolph P
- Morgan, Nathan N
- Taylor, Joseph R
- Zebo, Rachel
- Maxwell, Brad
- Moulin, Frederick
- Gordon, David A
- Robl, Jeffrey A
Publication details: ACS medicinal chemistry letters Dec 2018
In:
ACS medicinal chemistry letters vol. 9
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15.
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Discovery of Clinical Candidate 2-((2S,6S)-2-Phenyl-6-hydroxyadamantan-2-yl)-1-(3'-hydroxyazetidin-1-yl)ethanone [BMS-816336], an Orally Active Novel Selective 11β-Hydroxysteroid Dehydrogenase Type 1 Inhibitor. [electronic resource] by
- Ye, Xiang-Yang
- Chen, Stephanie Y
- Wu, Shung
- Yoon, David S
- Wang, Haixia
- Hong, Zhenqiu
- O'Connor, Stephen P
- Li, Jun
- Li, James J
- Kennedy, Lawrence J
- Walker, Steven J
- Nayeem, Akbar
- Sheriff, Steven
- Camac, Daniel M
- Ramamurthy, Vidyhashankar
- Morin, Paul E
- Zebo, Rachel
- Taylor, Joseph R
- Morgan, Nathan N
- Ponticiello, Randolph P
- Harrity, Thomas
- Apedo, Atsu
- Golla, Rajasree
- Seethala, Ramakrishna
- Wang, Mengmeng
- Harper, Timothy W
- Sleczka, Bogdan G
- He, Bin
- Kirby, Mark
- Leahy, David K
- Li, Jianqing
- Hanson, Ronald L
- Guo, Zhiwei
- Li, Yi-Xin
- DiMarco, John D
- Scaringe, Raymond
- Maxwell, Brad
- Moulin, Frederick
- Barrish, Joel C
- Gordon, David A
- Robl, Jeffrey A
Producer: 20170811
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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16.
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Discovery of an oxybenzylglycine based peroxisome proliferator activated receptor alpha selective agonist 2-((3-((2-(4-chlorophenyl)-5-methyloxazol-4-yl)methoxy)benzyl)(methoxycarbonyl)amino)acetic acid (BMS-687453). [electronic resource] by
- Li, Jun
- Kennedy, Lawrence J
- Shi, Yan
- Tao, Shiwei
- Ye, Xiang-Yang
- Chen, Stephanie Y
- Wang, Ying
- Hernández, Andrés S
- Wang, Wei
- Devasthale, Pratik V
- Chen, Sean
- Lai, Zhi
- Zhang, Hao
- Wu, Shung
- Smirk, Rebecca A
- Bolton, Scott A
- Ryono, Denis E
- Zhang, Huiping
- Lim, Ngiap-Kie
- Chen, Bang-Chi
- Locke, Kenneth T
- O'Malley, Kevin M
- Zhang, Litao
- Srivastava, Rai Ajit
- Miao, Bowman
- Meyers, Daniel S
- Monshizadegan, Hossain
- Search, Debra
- Grimm, Denise
- Zhang, Rongan
- Harrity, Thomas
- Kunselman, Lori K
- Cap, Michael
- Kadiyala, Pathanjali
- Hosagrahara, Vinayak
- Zhang, Lisa
- Xu, Carrie
- Li, Yi-Xin
- Muckelbauer, Jodi K
- Chang, Chiehying
- An, Yongmi
- Krystek, Stanley R
- Blanar, Michael A
- Zahler, Robert
- Mukherjee, Ranjan
- Cheng, Peter T W
- Tino, Joseph A
Producer: 20100510
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
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