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Pharmacokinetics and metabolism of AMG 232, a novel orally bioavailable inhibitor of the MDM2-p53 interaction, in rats, dogs and monkeys: in vitro-in vivo correlation. [electronic resource] by
- Ye, Qiuping
- Jiang, Min
- Huang, Wotang T
- Ling, Yun
- Olson, Steven H
- Sun, Daqing
- Xu, Guifen
- Yan, Xuelei
- Wong, Bradley K
- Jin, Lixia
Producer: 20160407
In:
Xenobiotica; the fate of foreign compounds in biological systems vol. 45
Availability: No items available.
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9.
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Synthesis, in Vitro Covalent Binding Evaluation, and Metabolism of (14)C-Labeled Inhibitors of 11β-HSD1. [electronic resource] by
- Sun, Daqing
- Ye, Qiuping
- Yan, Xuelei
- Rew, Yosup
- Fan, Peter
- He, Xiao
- Jiang, Min
- McMinn, Dustin L
- Monshouwer, Mario
- Tu, Hua
- Powers, Jay P
Producer: 20141121
In:
ACS medicinal chemistry letters vol. 5
Availability: No items available.
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10.
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Discovery and characterization of a potent and selective antagonist of melanin-concentrating hormone receptor 2. [electronic resource] by
- Chen, Xiaoqi
- Mihalic, Jeff
- Fan, Pingchen
- Liang, Lingming
- Lindstrom, Michelle
- Wong, Sylvia
- Ye, Qiuping
- Fu, Ying
- Jaen, Juan
- Chen, Jin-Long
- Dai, Kang
- Li, Leping
Producer: 20120803
In:
Bioorganic & medicinal chemistry letters vol. 22
Availability: No items available.
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11.
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Improvement of the synthesis and pharmacokinetic properties of chromenotriazolopyrimidine MDM2-p53 protein-protein inhibitors. [electronic resource] by
- Beck, Hilary P
- DeGraffenreid, Michael
- Fox, Brian
- Allen, John G
- Rew, Yosup
- Schneider, Stephen
- Saiki, Anne Y
- Yu, Dongyin
- Oliner, Jonathan D
- Salyers, Kevin
- Ye, Qiuping
- Olson, Steven
Producer: 20110815
In:
Bioorganic & medicinal chemistry letters vol. 21
Availability: No items available.
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12.
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Discovery and initial SAR of arylsulfonylpiperazine inhibitors of 11beta-hydroxysteroid dehydrogenase type 1 (11beta-HSD1). [electronic resource] by
- Sun, Daqing
- Wang, Zhulun
- Di, Yongmei
- Jaen, Juan C
- Labelle, Marc
- Ma, Ji
- Miao, Shichang
- Sudom, Athena
- Tang, Liang
- Tomooka, Craig S
- Tu, Hua
- Ursu, Stefania
- Walker, Nigel
- Yan, Xuelei
- Ye, Qiuping
- Powers, Jay P
Producer: 20080825
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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13.
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Discovery of potent, selective, and orally bioavailable inhibitors of interleukin-1 receptor-associate kinase-4. [electronic resource] by
- Wang, Zhulun
- Sun, Daqing
- Johnstone, Sheree
- Cao, Zhaodan
- Gao, Xiong
- Jaen, Juan C
- Liu, Jingqian
- Lively, Sarah
- Miao, Shichang
- Sudom, Athena
- Tomooka, Craig
- Walker, Nigel P C
- Wright, Matthew
- Yan, Xuelei
- Ye, Qiuping
- Powers, Jay P
Producer: 20161005
In:
Bioorganic & medicinal chemistry letters vol. 25
Availability: No items available.
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14.
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SAR and mode of action of novel non-nucleoside inhibitors of hepatitis C NS5b RNA polymerase. [electronic resource] by
- Powers, Jay P
- Piper, Derek E
- Li, Yang
- Mayorga, Veronica
- Anzola, John
- Chen, James M
- Jaen, Juan C
- Lee, Gary
- Liu, Jinqian
- Peterson, M Greg
- Tonn, George R
- Ye, Qiuping
- Walker, Nigel P C
- Wang, Zhulun
Producer: 20060329
In:
Journal of medicinal chemistry vol. 49
Availability: No items available.
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15.
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Discovery and optimization of piperidyl benzamide derivatives as a novel class of 11beta-HSD1 inhibitors. [electronic resource] by
- Rew, Yosup
- McMinn, Dustin L
- Wang, Zhulun
- He, Xiao
- Hungate, Randall W
- Jaen, Juan C
- Sudom, Athena
- Sun, Daqing
- Tu, Hua
- Ursu, Stefania
- Villemure, Elisia
- Walker, Nigel P C
- Yan, Xuelei
- Ye, Qiuping
- Powers, Jay P
Producer: 20090820
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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16.
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Discovery of a Potent Steroidal Glucocorticoid Receptor Antagonist with Enhanced Selectivity against the Progesterone and Androgen Receptors (OP-3633). [electronic resource] by
- Du, Xiaohui
- Eksterowicz, John
- Zhou, Haiying
- Rew, Yosup
- Zhu, Liusheng
- Yan, Xuelei
- Medina, Julio C
- Huang, Tom
- Chen, Xi
- Sutimantanapi, Dena
- Jahchan, Nadine
- Kong, Wayne
- Sun, Jessica
- Zavorotinskaya, Tatiana
- Ye, Qiuping
- Fantin, Valeria R
- Sun, Daqing
Producer: 20200615
In:
Journal of medicinal chemistry vol. 62
Availability: No items available.
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17.
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The MDM2 Inhibitor AMG 232 Demonstrates Robust Antitumor Efficacy and Potentiates the Activity of p53-Inducing Cytotoxic Agents. [electronic resource] by
- Canon, Jude
- Osgood, Tao
- Olson, Steven H
- Saiki, Anne Y
- Robertson, Rebecca
- Yu, Dongyin
- Eksterowicz, John
- Ye, Qiuping
- Jin, Lixia
- Chen, Ada
- Zhou, Jing
- Cordover, David
- Kaufman, Stephen
- Kendall, Richard
- Oliner, Jonathan D
- Coxon, Angela
- Radinsky, Robert
Producer: 20160316
In:
Molecular cancer therapeutics vol. 14
Availability: No items available.
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18.
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Synthesis and optimization of arylsulfonylpiperazines as a novel class of inhibitors of 11 beta-hydroxysteroid dehydrogenase type 1 (11 beta-HSD1). [electronic resource] by
- Sun, Daqing
- Wang, Zhulun
- Cardozo, Mario
- Choi, Rebekah
- Degraffenreid, Michael
- Di, Yongmei
- He, Xiao
- Jaen, Juan C
- Labelle, Marc
- Liu, Jinsong
- Ma, Ji
- Miao, Shichang
- Sudom, Athena
- Tang, Liang
- Tu, Hua
- Ursu, Stefania
- Walker, Nigel
- Yan, Xuelei
- Ye, Qiuping
- Powers, Jay P
Producer: 20090828
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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19.
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Discovery of a Potent and Selective Steroidal Glucocorticoid Receptor Antagonist (ORIC-101). [electronic resource] by
- Rew, Yosup
- Du, Xiaohui
- Eksterowicz, John
- Zhou, Haiying
- Jahchan, Nadine
- Zhu, Liusheng
- Yan, Xuelei
- Kawai, Hiroyuki
- McGee, Lawrence R
- Medina, Julio C
- Huang, Tom
- Chen, Chelsea
- Zavorotinskaya, Tatiana
- Sutimantanapi, Dena
- Waszczuk, Joanna
- Jackson, Erica
- Huang, Elizabeth
- Ye, Qiuping
- Fantin, Valeria R
- Sun, Daqing
Producer: 20191015
In:
Journal of medicinal chemistry vol. 61
Availability: No items available.
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20.
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Optimization of novel di-substituted cyclohexylbenzamide derivatives as potent 11 beta-HSD1 inhibitors. [electronic resource] by
- McMinn, Dustin L
- Rew, Yosup
- Sudom, Athena
- Caille, Seb
- Degraffenreid, Michael
- He, Xiao
- Hungate, Randall
- Jiang, Ben
- Jaen, Juan
- Julian, Lisa D
- Kaizerman, Jacob
- Novak, Perry
- Sun, Daqing
- Tu, Hua
- Ursu, Stefania
- Walker, Nigel P C
- Yan, Xuelei
- Ye, Qiuping
- Wang, Zhulun
- Powers, Jay P
Producer: 20090828
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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