Results
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A structure-guided optimization of pyrido[2,3-d]pyrimidin-7-ones as selective inhibitors of EGFR [electronic resource] by
- Yu, Lei
- Huang, Minhao
- Xu, Tianfeng
- Tong, Linjiang
- Yan, Xiao-E
- Zhang, Zhang
- Xu, Yong
- Yun, Caihong
- Xie, Hua
- Ding, Ke
- Lu, Xiaoyun
Producer: 20170222
In:
European journal of medicinal chemistry vol. 126
Availability: No items available.
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6.
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Discovery of 4-((N-(2-(dimethylamino)ethyl)acrylamido)methyl)-N-(4-methyl-3-((4-(pyridin-3-yl)pyrimidin-2-yl)amino)phenyl)benzamide (CHMFL-PDGFR-159) as a highly selective type II PDGFRα kinase inhibitor for PDGFRα driving chronic eosinophilic leukemia. [electronic resource] by
- Wang, Qiang
- Liu, Feiyang
- Qi, Shuang
- Qi, Ziping
- Yan, Xiao-E
- Wang, Beilei
- Wang, Aoli
- Wang, Wei
- Chen, Cheng
- Liu, Xiaochuan
- Jiang, Zongru
- Hu, Zhenquan
- Wang, Li
- Wang, Wenchao
- Ren, Tao
- Zhang, Shanchun
- Yun, Cai-Hong
- Liu, Qingsong
- Liu, Jing
Producer: 20180426
In:
European journal of medicinal chemistry vol. 150
Availability: No items available.
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7.
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Discovery and characterization of a novel irreversible EGFR mutants selective and potent kinase inhibitor CHMFL-EGFR-26 with a distinct binding mode. [electronic resource] by
- Hu, Chen
- Wang, Aoli
- Wu, Hong
- Qi, Ziping
- Li, Xixiang
- Yan, Xiao-E
- Chen, Cheng
- Yu, Kailin
- Zou, Fengming
- Wang, Wenchao
- Wang, Wei
- Wu, Jiaxin
- Liu, Juan
- Wang, Beilei
- Wang, Li
- Ren, Tao
- Zhang, Shanchun
- Yun, Cai-Hong
- Liu, Jing
- Liu, Qingsong
Producer: 20170929
In:
Oncotarget vol. 8
Availability: No items available.
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8.
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Discovery of (R)-1-(3-(4-Amino-3-(3-chloro-4-(pyridin-2-ylmethoxy)phenyl)-1H-pyrazolo[3,4-d]pyrimidin-1-yl)piperidin-1-yl)prop-2-en-1-one (CHMFL-EGFR-202) as a Novel Irreversible EGFR Mutant Kinase Inhibitor with a Distinct Binding Mode. [electronic resource] by
- Wang, Aoli
- Li, Xixiang
- Wu, Hong
- Zou, Fengming
- Yan, Xiao-E
- Chen, Cheng
- Hu, Chen
- Yu, Kailin
- Wang, Wenchao
- Zhao, Peng
- Wu, Jiaxin
- Qi, Ziping
- Wang, Wei
- Wang, Beilei
- Wang, Li
- Ren, Tao
- Zhang, Shanchun
- Yun, Cai-Hong
- Liu, Jing
- Liu, Qingsong
Producer: 20170424
In:
Journal of medicinal chemistry vol. 60
Availability: No items available.
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9.
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Ibrutinib targets mutant-EGFR kinase with a distinct binding conformation. [electronic resource] by
- Wang, Aoli
- Yan, Xiao-E
- Wu, Hong
- Wang, Wenchao
- Hu, Chen
- Chen, Cheng
- Zhao, Zheng
- Zhao, Peng
- Li, Xixiang
- Wang, Li
- Wang, Beilei
- Ye, Zi
- Wang, Jinhua
- Wang, Chu
- Zhang, Wei
- Gray, Nathanael S
- Weisberg, Ellen L
- Chen, Liang
- Liu, Jing
- Yun, Cai-Hong
- Liu, Qingsong
Producer: 20180213
In:
Oncotarget vol. 7
Availability: No items available.
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10.
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Ibrutinib selectively and irreversibly targets EGFR (L858R, Del19) mutant but is moderately resistant to EGFR (T790M) mutant NSCLC Cells. [electronic resource] by
- Wu, Hong
- Wang, Aoli
- Zhang, Wei
- Wang, Beilei
- Chen, Cheng
- Wang, Wenchao
- Hu, Chen
- Ye, Zi
- Zhao, Zheng
- Wang, Li
- Li, Xixiang
- Yu, Kailin
- Liu, Juan
- Wu, Jiaxin
- Yan, Xiao-E
- Zhao, Peng
- Wang, Jinhua
- Wang, Chu
- Weisberg, Ellen L
- Gray, Nathanael S
- Yun, Cai-Hong
- Liu, Jing
- Chen, Liang
- Liu, Qingsong
Producer: 20160823
In:
Oncotarget vol. 6
Availability: No items available.
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