Optimization of 4-phenylamino-3-quinolinecarbonitriles as potent inhibitors of Src kinase activity. [electronic resource]
Producer: 20011207Description: 3965-77 p. digitalISSN:- 0022-2623
- Animals
- Antineoplastic Agents -- chemical synthesis
- Cell Division -- drug effects
- Cell Line, Transformed
- Enzyme Inhibitors -- chemical synthesis
- Female
- Fibroblasts -- metabolism
- Humans
- Immunoblotting
- Mice
- Mice, Inbred BALB C
- Mice, Nude
- Nitriles -- chemical synthesis
- Phosphorylation
- Piperazines -- chemical synthesis
- Quinolines -- chemical synthesis
- Structure-Activity Relationship
- Tumor Cells, Cultured
- Tyrosine -- metabolism
- Xenograft Model Antitumor Assays
- src-Family Kinases -- antagonists & inhibitors
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Publication Type: Journal Article
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