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  2. Details for: Optimization of 4-phenylamino-3-quinolinecarbonitriles as potent inhibitors of Src kinase activity.
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Optimization of 4-phenylamino-3-quinolinecarbonitriles as potent inhibitors of Src kinase activity. [electronic resource]

By:
  • Boschelli, D H
Contributor(s):
  • Ye, F
  • Wang, Y D
  • Dutia, M
  • Johnson, S L
  • Wu, B
  • Miller, K
  • Powell, D W
  • Yaczko, D
  • Young, M
  • Tischler, M
  • Arndt, K
  • Discafani, C
  • Etienne, C
  • Gibbons, J
  • Grod, J
  • Lucas, J
  • Weber, J M
  • Boschelli, F
Producer: 20011207Description: 3965-77 p. digitalISSN:
  • 0022-2623
Subject(s):
  • Animals
  • Antineoplastic Agents -- chemical synthesis
  • Cell Division -- drug effects
  • Cell Line, Transformed
  • Enzyme Inhibitors -- chemical synthesis
  • Female
  • Fibroblasts -- metabolism
  • Humans
  • Immunoblotting
  • Mice
  • Mice, Inbred BALB C
  • Mice, Nude
  • Nitriles -- chemical synthesis
  • Phosphorylation
  • Piperazines -- chemical synthesis
  • Quinolines -- chemical synthesis
  • Structure-Activity Relationship
  • Tumor Cells, Cultured
  • Tyrosine -- metabolism
  • Xenograft Model Antitumor Assays
  • src-Family Kinases -- antagonists & inhibitors
Online resources:
  • Available from publisher's website
In: Journal of medicinal chemistry vol. 44
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Publication Type: Journal Article

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Optimization of 4-phenylamino-3-quinolinecarbonitriles as potent inhibitors of Src kinase activity.

APA

Boschelli D. H., Ye F., Wang Y. D., Dutia M., Johnson S. L., Wu B., Miller K., Powell D. W., Yaczko D., Young M., Tischler M., Arndt K., Discafani C., Etienne C., Gibbons J., Grod J., Lucas J., Weber J. M. & Boschelli F. (20011207). Optimization of 4-phenylamino-3-quinolinecarbonitriles as potent inhibitors of Src kinase activity. : Journal of medicinal chemistry.

Chicago

Boschelli D H, Ye F, Wang Y D, Dutia M, Johnson S L, Wu B, Miller K, Powell D W, Yaczko D, Young M, Tischler M, Arndt K, Discafani C, Etienne C, Gibbons J, Grod J, Lucas J, Weber J M and Boschelli F. 20011207. Optimization of 4-phenylamino-3-quinolinecarbonitriles as potent inhibitors of Src kinase activity. : Journal of medicinal chemistry.

Harvard

Boschelli D. H., Ye F., Wang Y. D., Dutia M., Johnson S. L., Wu B., Miller K., Powell D. W., Yaczko D., Young M., Tischler M., Arndt K., Discafani C., Etienne C., Gibbons J., Grod J., Lucas J., Weber J. M. and Boschelli F. (20011207). Optimization of 4-phenylamino-3-quinolinecarbonitriles as potent inhibitors of Src kinase activity. : Journal of medicinal chemistry.

MLA

Boschelli D H, Ye F, Wang Y D, Dutia M, Johnson S L, Wu B, Miller K, Powell D W, Yaczko D, Young M, Tischler M, Arndt K, Discafani C, Etienne C, Gibbons J, Grod J, Lucas J, Weber J M and Boschelli F. Optimization of 4-phenylamino-3-quinolinecarbonitriles as potent inhibitors of Src kinase activity. : Journal of medicinal chemistry. 20011207.

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