Results
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1.
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Hydroxyethylamine-based inhibitors of BACE1: P₁-P₃ macrocyclization can improve potency, selectivity, and cell activity. [electronic resource] by
- Pennington, Lewis D
- Whittington, Douglas A
- Bartberger, Michael D
- Jordan, Steven R
- Monenschein, Holger
- Nguyen, Thomas T
- Yang, Bryant H
- Xue, Qiufen M
- Vounatsos, Filisaty
- Wahl, Robert C
- Chen, Kui
- Wood, Stephen
- Citron, Martin
- Patel, Vinod F
- Hitchcock, Stephen A
- Zhong, Wenge
Producer: 20140124
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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2.
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Inhibitors of human immunodeficiency virus type 1 (HIV-1) attachment. 12. Structure-activity relationships associated with 4-fluoro-6-azaindole derivatives leading to the identification of 1-(4-benzoylpiperazin-1-yl)-2-(4-fluoro-7-[1,2,3]triazol-1-yl-1h-pyrrolo[2,3-c]pyridin-3-yl)ethane-1,2-dione (BMS-585248). [electronic resource] by
- Regueiro-Ren, Alicia
- Xue, Qiufen M
- Swidorski, Jacob J
- Gong, Yi-Fei
- Mathew, Marina
- Parker, Dawn D
- Yang, Zheng
- Eggers, Betsy
- D'Arienzo, Celia
- Sun, Yongnian
- Malinowski, Jacek
- Gao, Qi
- Wu, Dedong
- Langley, David R
- Colonno, Richard J
- Chien, Caly
- Grasela, Dennis M
- Zheng, Ming
- Lin, Pin-Fang
- Meanwell, Nicholas A
- Kadow, John F
Producer: 20130731
In:
Journal of medicinal chemistry vol. 56
Availability: No items available.
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3.
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Design and preparation of a potent series of hydroxyethylamine containing β-secretase inhibitors that demonstrate robust reduction of central β-amyloid. [electronic resource] by
- Weiss, Matthew M
- Williamson, Toni
- Babu-Khan, Safura
- Bartberger, Michael D
- Brown, James
- Chen, Kui
- Cheng, Yuan
- Citron, Martin
- Croghan, Michael D
- Dineen, Thomas A
- Esmay, Joel
- Graceffa, Russell F
- Harried, Scott S
- Hickman, Dean
- Hitchcock, Stephen A
- Horne, Daniel B
- Huang, Hongbing
- Imbeah-Ampiah, Ronke
- Judd, Ted
- Kaller, Matthew R
- Kreiman, Charles R
- La, Daniel S
- Li, Vivian
- Lopez, Patricia
- Louie, Steven
- Monenschein, Holger
- Nguyen, Thomas T
- Pennington, Lewis D
- Rattan, Claire
- San Miguel, Tisha
- Sickmier, E Allen
- Wahl, Robert C
- Wen, Paul H
- Wood, Stephen
- Xue, Qiufen
- Yang, Bryant H
- Patel, Vinod F
- Zhong, Wenge
Producer: 20130226
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
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4.
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Design and synthesis of potent, orally efficacious hydroxyethylamine derived β-site amyloid precursor protein cleaving enzyme (BACE1) inhibitors. [electronic resource] by
- Dineen, Thomas A
- Weiss, Matthew M
- Williamson, Toni
- Acton, Paul
- Babu-Khan, Safura
- Bartberger, Michael D
- Brown, James
- Chen, Kui
- Cheng, Yuan
- Citron, Martin
- Croghan, Michael D
- Dunn, Robert T
- Esmay, Joel
- Graceffa, Russell F
- Harried, Scott S
- Hickman, Dean
- Hitchcock, Stephen A
- Horne, Daniel B
- Huang, Hongbing
- Imbeah-Ampiah, Ronke
- Judd, Ted
- Kaller, Matthew R
- Kreiman, Charles R
- La, Daniel S
- Li, Vivian
- Lopez, Patricia
- Louie, Steven
- Monenschein, Holger
- Nguyen, Thomas T
- Pennington, Lewis D
- San Miguel, Tisha
- Sickmier, E Allen
- Vargas, Hugo M
- Wahl, Robert C
- Wen, Paul H
- Whittington, Douglas A
- Wood, Stephen
- Xue, Qiufen
- Yang, Bryant H
- Patel, Vinod F
- Zhong, Wenge
Producer: 20130226
In:
Journal of medicinal chemistry vol. 55
Availability: No items available.
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