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Synthesis and SAR of p38alpha MAP kinase inhibitors based on heterobicyclic scaffolds. [electronic resource] by
- Murali Dhar, T G
- Wrobleski, Stephen T
- Lin, Shuqun
- Furch, Joseph A
- Nirschl, David S
- Fan, Yi
- Todderud, Gordon
- Pitt, Sidney
- Doweyko, Arthur M
- Sack, John S
- Mathur, Arvind
- McKinnon, Murray
- Barrish, Joel C
- Dodd, John H
- Schieven, Gary L
- Leftheris, Katerina
Producer: 20071227
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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8.
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Rational design and synthesis of an orally active indolopyridone as a novel conformationally constrained cannabinoid ligand possessing antiinflammatory properties. [electronic resource] by
- Wrobleski, Stephen T
- Chen, Ping
- Hynes, John
- Lin, Shuqun
- Norris, Derek J
- Pandit, Chennagiri R
- Spergel, Steven
- Wu, Hong
- Tokarski, John S
- Chen, Xiaorong
- Gillooly, Kathleen M
- Kiener, Peter A
- McIntyre, Kim W
- Patil-Koota, Vina
- Shuster, David J
- Turk, Lori A
- Yang, Guchen
- Leftheris, Katerina
Producer: 20030623
In:
Journal of medicinal chemistry vol. 46
Availability: No items available.
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9.
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Utilization of a nitrogen-sulfur nonbonding interaction in the design of new 2-aminothiazol-5-yl-pyrimidines as p38α MAP kinase inhibitors. [electronic resource] by
- Lin, Shuqun
- Wrobleski, Stephen T
- Hynes, John
- Pitt, Sidney
- Zhang, Rosemary
- Fan, Yi
- Doweyko, Arthur M
- Kish, Kevin F
- Sack, John S
- Malley, Mary F
- Kiefer, Susan E
- Newitt, John A
- McKinnon, Murray
- Trzaskos, James
- Barrish, Joel C
- Dodd, John H
- Schieven, Gary L
- Leftheris, Katerina
Producer: 20110224
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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10.
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5-Cyanopyrimidine derivatives as a novel class of potent, selective, and orally active inhibitors of p38alpha MAP kinase. [electronic resource] by
- Liu, Chunjian
- Wrobleski, Stephen T
- Lin, James
- Ahmed, Gulzar
- Metzger, Axel
- Wityak, John
- Gillooly, Kathleen M
- Shuster, David J
- McIntyre, Kim W
- Pitt, Sidney
- Shen, Ding Ren
- Zhang, Rosemary F
- Zhang, Hongjian
- Doweyko, Arthur M
- Diller, David
- Henderson, Ian
- Barrish, Joel C
- Dodd, John H
- Schieven, Gary L
- Leftheris, Katerina
Producer: 20051128
In:
Journal of medicinal chemistry vol. 48
Availability: No items available.
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11.
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Synthesis and SAR of new pyrrolo[2,1-f][1,2,4]triazines as potent p38 alpha MAP kinase inhibitors. [electronic resource] by
- Wrobleski, Stephen T
- Lin, Shuqun
- Hynes, John
- Wu, Hong
- Pitt, Sidney
- Shen, Ding Ren
- Zhang, Rosemary
- Gillooly, Kathleen M
- Shuster, David J
- McIntyre, Kim W
- Doweyko, Arthur M
- Kish, Kevin F
- Tredup, Jeffrey A
- Duke, Gerald J
- Sack, John S
- McKinnon, Murray
- Dodd, John
- Barrish, Joel C
- Schieven, Gary L
- Leftheris, Katerina
Producer: 20080516
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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12.
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The identification of novel p38α isoform selective kinase inhibitors having an unprecedented p38α binding mode. [electronic resource] by
- Wrobleski, Stephen T
- Lin, Shuqun
- Dhar, T G Murali
- Dyckman, Alaric J
- Li, Tianle
- Pitt, Sidney
- Zhang, Rosemary
- Fan, Yi
- Doweyko, Arthur M
- Tokarski, John S
- Kish, Kevin F
- Kiefer, Susan E
- Sack, John S
- Newitt, John A
- Witmer, Mark R
- McKinnon, Murray
- Barrish, Joel C
- Dodd, John H
- Schieven, Gary L
- Leftheris, Katerina
Producer: 20140121
In:
Bioorganic & medicinal chemistry letters vol. 23
Availability: No items available.
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13.
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Discovery of highly potent, selective, covalent inhibitors of JAK3. [electronic resource] by
- Kempson, James
- Ovalle, Damaso
- Guo, Junqing
- Wrobleski, Stephen T
- Lin, Shuqun
- Spergel, Steven H
- Duan, James J-W
- Jiang, Bin
- Lu, Zhonghui
- Das, Jagabandhu
- Yang, Bingwei V
- Hynes, John
- Wu, Hong
- Tokarski, John
- Sack, John S
- Khan, Javed
- Schieven, Gary
- Blatt, Yuval
- Chaudhry, Charu
- Salter-Cid, Luisa M
- Fura, Aberra
- Barrish, Joel C
- Carter, Percy H
- Pitts, William J
Producer: 20171103
In:
Bioorganic & medicinal chemistry letters vol. 27
Availability: No items available.
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14.
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Discovery of potent and efficacious pyrrolopyridazines as dual JAK1/3 inhibitors. [electronic resource] by
- Hynes, John
- Wu, Hong
- Kempson, James
- Duan, James J-W
- Lu, Zhonghui
- Jiang, Bin
- Stachura, Sylwia
- Tokarski, John S
- Sack, John S
- Khan, Javed A
- Lippy, Jonathan S
- Zhang, Rosemary F
- Pitt, Sidney
- Shen, Guoxiang
- Gillooly, Kate
- McIntyre, Kim
- Carter, Percy H
- Barrish, Joel C
- Nadler, Steven G
- Salter-Cid, Luisa M
- Fura, Aberra
- Schieven, Gary L
- Pitts, William J
- Wrobleski, Stephen T
Producer: 20170914
In:
Bioorganic & medicinal chemistry letters vol. 27
Availability: No items available.
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15.
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Identification of [electronic resource] by
- Moslin, Ryan
- Zhang, Yanlei
- Wrobleski, Stephen T
- Lin, Shuqun
- Mertzman, Michael
- Spergel, Steven
- Tokarski, John S
- Strnad, Joann
- Gillooly, Kathleen
- McIntyre, Kim W
- Zupa-Fernandez, Adriana
- Cheng, Lihong
- Sun, Huadong
- Chaudhry, Charu
- Huang, Christine
- D'Arienzo, Celia
- Heimrich, Elizabeth
- Yang, Xiaoxia
- Muckelbauer, Jodi K
- Chang, ChiehYing
- Tredup, Jeffrey
- Mulligan, Dawn
- Xie, Dianlin
- Aranibar, Nelly
- Chiney, Manoj
- Burke, James R
- Lombardo, Louis
- Carter, Percy H
- Weinstein, David S
Producer: 20200706
In:
Journal of medicinal chemistry vol. 62
Availability: No items available.
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16.
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Discovery of ((4-(5-(Cyclopropylcarbamoyl)-2-methylphenylamino)-5-methylpyrrolo[1,2-f][1,2,4]triazine-6-carbonyl)(propyl)carbamoyloxy)methyl-2-(4-(phosphonooxy)phenyl)acetate (BMS-751324), a Clinical Prodrug of p38α MAP Kinase Inhibitor. [electronic resource] by
- Liu, Chunjian
- Lin, James
- Hynes, John
- Wu, Hong
- Wrobleski, Stephen T
- Lin, Shuqun
- Dhar, T G Murali
- Vrudhula, Vivekananda M
- Sun, Jung-Hui
- Chao, Sam
- Zhao, Rulin
- Wang, Bei
- Chen, Bang-Chi
- Everlof, Gerry
- Gesenberg, Christoph
- Zhang, Hongjian
- Marathe, Punit H
- McIntyre, Kim W
- Taylor, Tracy L
- Gillooly, Kathleen
- Shuster, David J
- McKinnon, Murray
- Dodd, John H
- Barrish, Joel C
- Schieven, Gary L
- Leftheris, Katerina
Producer: 20160504
In:
Journal of medicinal chemistry vol. 58
Availability: No items available.
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17.
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Discovery of a JAK1/3 Inhibitor and Use of a Prodrug To Demonstrate Efficacy in a Model of Rheumatoid Arthritis. [electronic resource] by
- Spergel, Steven H
- Mertzman, Michael E
- Kempson, James
- Guo, Junqing
- Stachura, Sylwia
- Haque, Lauren
- Lippy, Jonathan S
- Zhang, Rosemary F
- Galella, Michael
- Pitt, Sidney
- Shen, Guoxiang
- Fura, Aberra
- Gillooly, Kathleen
- McIntyre, Kim W
- Tang, Vicky
- Tokarski, John
- Sack, John S
- Khan, Javed
- Carter, Percy H
- Barrish, Joel C
- Nadler, Steven G
- Salter-Cid, Luisa M
- Schieven, Gary L
- Wrobleski, Stephen T
- Pitts, William J
Publication details: ACS medicinal chemistry letters Mar 2019
In:
ACS medicinal chemistry letters vol. 10
Availability: No items available.
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18.
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Discovery of pyrrolo[1,2-b]pyridazine-3-carboxamides as Janus kinase (JAK) inhibitors. [electronic resource] by
- Duan, James J-W
- Lu, Zhonghui
- Jiang, Bin
- Yang, Bingwei V
- Doweyko, Lidia M
- Nirschl, David S
- Haque, Lauren E
- Lin, Shuqun
- Brown, Gregory
- Hynes, John
- Tokarski, John S
- Sack, John S
- Khan, Javed
- Lippy, Jonathan S
- Zhang, Rosemary F
- Pitt, Sidney
- Shen, Guoxiang
- Pitts, William J
- Carter, Percy H
- Barrish, Joel C
- Nadler, Steven G
- Salter-Cid, Luisa M
- McKinnon, Murray
- Fura, Aberra
- Schieven, Gary L
- Wrobleski, Stephen T
Producer: 20150804
In:
Bioorganic & medicinal chemistry letters vol. 24
Availability: No items available.
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19.
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Design, synthesis, and anti-inflammatory properties of orally active 4-(phenylamino)-pyrrolo[2,1-f][1,2,4]triazine p38alpha mitogen-activated protein kinase inhibitors. [electronic resource] by
- Hynes, John
- Dyckman, Alaric J
- Lin, Shuqun
- Wrobleski, Stephen T
- Wu, Hong
- Gillooly, Kathleen M
- Kanner, Steven B
- Lonial, Herinder
- Loo, Derek
- McIntyre, Kim W
- Pitt, Sidney
- Shen, Ding Ren
- Shuster, David J
- Yang, Xiaoxia
- Zhang, Rosemary
- Behnia, Kamelia
- Zhang, Hongjian
- Marathe, Punit H
- Doweyko, Arthur M
- Tokarski, John S
- Sack, John S
- Pokross, Matthew
- Kiefer, Susan E
- Newitt, John A
- Barrish, Joel C
- Dodd, John
- Schieven, Gary L
- Leftheris, Katerina
Producer: 20080227
In:
Journal of medicinal chemistry vol. 51
Availability: No items available.
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20.
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Autoimmune pathways in mice and humans are blocked by pharmacological stabilization of the TYK2 pseudokinase domain. [electronic resource] by
- Burke, James R
- Cheng, Lihong
- Gillooly, Kathleen M
- Strnad, Joann
- Zupa-Fernandez, Adriana
- Catlett, Ian M
- Zhang, Yifan
- Heimrich, Elizabeth M
- McIntyre, Kim W
- Cunningham, Mark D
- Carman, Julie A
- Zhou, Xiadi
- Banas, Dana
- Chaudhry, Charu
- Li, Sha
- D'Arienzo, Celia
- Chimalakonda, Anjaneya
- Yang, XiaoXia
- Xie, Jenny H
- Pang, Jian
- Zhao, Qihong
- Rose, Shawn M
- Huang, Jinwen
- Moslin, Ryan M
- Wrobleski, Stephen T
- Weinstein, David S
- Salter-Cid, Luisa M
Producer: 20200727
In:
Science translational medicine vol. 11
Availability: No items available.
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