Results
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2.
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B-Raf kinase inhibitors: hit enrichment through scaffold hopping. [electronic resource] by
- Gopalsamy, Ariamala
- Shi, Mengxiao
- Hu, Yongbo
- Lee, Frederick
- Feldberg, Larry
- Frommer, Eileen
- Kim, Steven
- Collins, Karen
- Wojciechowicz, Donald
- Mallon, Robert
Producer: 20100812
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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3.
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Identification of pyrazolo[1,5-a]pyrimidine-3-carboxylates as B-Raf kinase inhibitors. [electronic resource] by
- Gopalsamy, Ariamala
- Ciszewski, Greg
- Hu, Yongbo
- Lee, Frederick
- Feldberg, Larry
- Frommer, Eileen
- Kim, Steven
- Collins, Karen
- Wojciechowicz, Donald
- Mallon, Robert
Producer: 20090629
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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4.
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Discovery of highly potent and selective type I B-Raf kinase inhibitors. [electronic resource] by
- Wang, Xiaolun
- Berger, Dan M
- Salaski, Edward J
- Torres, Nancy
- Hu, Yongbo
- Levin, Jeremy I
- Powell, Dennis
- Wojciechowicz, Donald
- Collins, Karen
- Frommer, Eileen
Producer: 20100119
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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5.
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Hit to lead optimization of pyrazolo[1,5-a]pyrimidines as B-Raf kinase inhibitors. [electronic resource] by
- Gopalsamy, Ariamala
- Ciszewski, Greg
- Shi, Mengxiao
- Berger, Dan
- Hu, Yongbo
- Lee, Frederick
- Feldberg, Larry
- Frommer, Eileen
- Kim, Steven
- Collins, Karen
- Wojciechowicz, Donald
- Mallon, Robert
Producer: 20100209
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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6.
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4-Anilino-7-alkenylquinoline-3-carbonitriles as potent MEK1 kinase inhibitors. [electronic resource] by
- Berger, Dan M
- Dutia, Minu
- Powell, Dennis
- Floyd, Middleton B
- Torres, Nancy
- Mallon, Robert
- Wojciechowicz, Donald
- Kim, Steven
- Feldberg, Larry
- Collins, Karen
- Chaudhary, Inder
Producer: 20081215
In:
Bioorganic & medicinal chemistry vol. 16
Availability: No items available.
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7.
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Identification of 4-anilino-3-quinolinecarbonitrile inhibitors of mitogen-activated protein/extracellular signal-regulated kinase 1 kinase. [electronic resource] by
- Mallon, Robert
- Feldberg, Larry
- Kim, Steven
- Collins, Karen
- Wojciechowicz, Donald
- Kohler, Constance
- Kovacs, Diana
- Discafani, Carolyn
- Zhang, Nan
- Wu, Biqi
- Floyd, Brawner
- Powell, Dennis
- Berger, Dan
Producer: 20050118
In:
Molecular cancer therapeutics vol. 3
Availability: No items available.
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8.
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Aldisine alkaloids from the Philippine sponge Stylissa massa are potent inhibitors of mitogen-activated protein kinase kinase-1 (MEK-1). [electronic resource] by
- Tasdemir, Deniz
- Mallon, Robert
- Greenstein, Michael
- Feldberg, Larry R
- Kim, Steven C
- Collins, Karen
- Wojciechowicz, Donald
- Mangalindan, Gina C
- Concepción, Gisela P
- Harper, Mary Kay
- Ireland, Chris M
Producer: 20020207
In:
Journal of medicinal chemistry vol. 45
Availability: No items available.
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9.
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Indazolylpyrazolopyrimidine as highly potent B-Raf inhibitors with in vivo activity. [electronic resource] by
- Wang, Xiaolun
- Berger, Dan M
- Salaski, Edward J
- Torres, Nancy
- Dutia, Minu
- Hanna, Cilien
- Hu, Yongbo
- Levin, Jeremy I
- Powell, Dennis
- Wojciechowicz, Donald
- Collins, Karen
- Frommer, Eileen
- Lucas, Judy
Producer: 20101228
In:
Journal of medicinal chemistry vol. 53
Availability: No items available.
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10.
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Epithelial tissue hyperplasia induced by the RAF inhibitor PF-04880594 is attenuated by a clinically well-tolerated dose of the MEK inhibitor PD-0325901. [electronic resource] by
- Torti, Vince R
- Wojciechowicz, Donald
- Hu, Wenyue
- John-Baptiste, Annette
- Evering, Winston
- Troche, Gabriel
- Marroquin, Lisa D
- Smeal, Tod
- Yamazaki, Shinji
- Palmer, Cynthia L
- Burns-Naas, Leigh Ann
- Bagrodia, Shubha
Producer: 20130708
In:
Molecular cancer therapeutics vol. 11
Availability: No items available.
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11.
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Non-hinge-binding pyrazolo[1,5-a]pyrimidines as potent B-Raf kinase inhibitors. [electronic resource] by
- Berger, Dan M
- Torres, Nancy
- Dutia, Minu
- Powell, Dennis
- Ciszewski, Greg
- Gopalsamy, Ariamala
- Levin, Jeremy I
- Kim, Kyung-Hee
- Xu, Weixin
- Wilhelm, James
- Hu, YongBo
- Collins, Karen
- Feldberg, Larry
- Kim, Steven
- Frommer, Eileen
- Wojciechowicz, Donald
- Mallon, Robert
Producer: 20100119
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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12.
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Synthesis and evaluation of 4-anilino-6,7-dialkoxy-3-quinolinecarbonitriles as inhibitors of kinases of the Ras-MAPK signaling cascade. [electronic resource] by
- Berger, Dan
- Dutia, Minu
- Powell, Dennis
- Wu, Biqi
- Wissner, Allan
- Boschelli, Diane H
- Floyd, M Brawner
- Zhang, Nan
- Torres, Nancy
- Levin, Jeremy
- Du, Xuemei
- Wojciechowicz, Donald
- Discafani, Carolyn
- Kohler, Constance
- Kim, Steven C
- Feldberg, Larry R
- Collins, Karen
- Mallon, Robert
Producer: 20040521
In:
Bioorganic & medicinal chemistry letters vol. 13
Availability: No items available.
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13.
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Novel pyrazolopyrimidines as highly potent B-Raf inhibitors. [electronic resource] by
- Di Grandi, Martin J
- Berger, Dan M
- Hopper, Darrin W
- Zhang, Chunchun
- Dutia, Minu
- Dunnick, Alejandro L
- Torres, Nancy
- Levin, Jeremy I
- Diamantidis, George
- Zapf, Christoph W
- Bloom, Jonathan D
- Hu, YongBo
- Powell, Dennis
- Wojciechowicz, Donald
- Collins, Karen
- Frommer, Eileen
Producer: 20100209
In:
Bioorganic & medicinal chemistry letters vol. 19
Availability: No items available.
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