Results
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1.
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Imidazole moiety replacements in the 3-(1H-benzo[d]imidazol-2-yl)pyridin-2(1H)-one inhibitors of insulin-like growth factor receptor-1 (IGF-1R) to improve cytochrome P450 profile. [electronic resource] by
- Velaparthi, Upender
- Liu, Peiying
- Balasubramanian, Balu
- Carboni, Joan
- Attar, Ricardo
- Gottardis, Marco
- Li, Aixin
- Greer, Ann
- Zoeckler, Mary
- Wittman, Mark D
- Vyas, Dolatrai
Producer: 20070807
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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2.
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3.
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2-(1H-Imidazol-4-yl)ethanamine and 2-(1H-pyrazol-1-yl)ethanamine side chain variants of the IGF-1R inhibitor BMS-536924. [electronic resource] by
- Saulnier, Mark G
- Frennesson, David B
- Wittman, Mark D
- Zimmermann, Kurt
- Velaparthi, Upender
- Langley, David R
- Struzynski, Charles
- Sang, Xiaopeng
- Carboni, Joan
- Li, Aixin
- Greer, Ann
- Yang, Zheng
- Balimane, Praveen
- Gottardis, Marco
- Attar, Ricardo
- Vyas, Dolatrai
Producer: 20080519
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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4.
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Novel 1H-(benzimidazol-2-yl)-1H-pyridin-2-one inhibitors of insulin-like growth factor I (IGF-1R) kinase. [electronic resource] by
- Wittman, Mark D
- Balasubramanian, Balu
- Stoffan, Karen
- Velaparthi, Upender
- Liu, Pieying
- Krishnanathan, Subramaniam
- Carboni, Joan
- Li, Aixin
- Greer, Ann
- Attar, Ricardo
- Gottardis, Marco
- Chang, Chiehying
- Jacobson, Bruce
- Sun, Yax
- Hansel, Steven
- Zoeckler, Mary
- Vyas, Dolatrai M
Producer: 20070413
In:
Bioorganic & medicinal chemistry letters vol. 17
Availability: No items available.
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5.
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Insulin-like growth factor-1 receptor (IGF-1R) kinase inhibitors: SAR of a series of 3-[6-(4-substituted-piperazin-1-yl)-4-methyl-1H-benzimidazol-2-yl]-1H-pyridine-2-one. [electronic resource] by
- Velaparthi, Upender
- Saulnier, Mark G
- Wittman, Mark D
- Liu, Peiying
- Frennesson, David B
- Zimmermann, Kurt
- Carboni, Joan M
- Gottardis, Marco
- Li, Aixin
- Greer, Ann
- Clarke, Wendy
- Yang, Zheng
- Menard, Krista
- Lee, Francis Y
- Trainor, George
- Vyas, Dolatrai
Producer: 20100802
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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6.
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Balancing oral exposure with Cyp3A4 inhibition in benzimidazole-based IGF-IR inhibitors. [electronic resource] by
- Zimmermann, Kurt
- Wittman, Mark D
- Saulnier, Mark G
- Velaparthi, Upender
- Langley, David R
- Sang, Xiaopeng
- Frennesson, David
- Carboni, Joan
- Li, Aixin
- Greer, Ann
- Gottardis, Marco
- Attar, Ricardo M
- Yang, Zheng
- Balimane, Praveen
- Discenza, Lorell N
- Vyas, Dolatrai
Producer: 20081117
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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7.
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SAR of PXR transactivation in benzimidazole-based IGF-1R kinase inhibitors. [electronic resource] by
- Zimmermann, Kurt
- Wittman, Mark D
- Saulnier, Mark G
- Velaparthi, Upender
- Sang, Xiaopeng
- Frennesson, David B
- Struzynski, Charles
- Seitz, Steven P
- He, Liqi
- Carboni, Joan M
- Li, Aixin
- Greer, Ann F
- Gottardis, Marco
- Attar, Ricardo M
- Yang, Zheng
- Balimane, Praveen
- Discenza, Lorell N
- Lee, Francis Y
- Sinz, Michael
- Kim, Sean
- Vyas, Dolatrai
Producer: 20100527
In:
Bioorganic & medicinal chemistry letters vol. 20
Availability: No items available.
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8.
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Discovery of a 2,4-disubstituted pyrrolo[1,2-f][1,2,4]triazine inhibitor (BMS-754807) of insulin-like growth factor receptor (IGF-1R) kinase in clinical development. [electronic resource] by
- Wittman, Mark D
- Carboni, Joan M
- Yang, Zheng
- Lee, Francis Y
- Antman, Melissa
- Attar, Ricardo
- Balimane, Praveen
- Chang, Chiehying
- Chen, Cliff
- Discenza, Lorell
- Frennesson, David
- Gottardis, Marco M
- Greer, Ann
- Hurlburt, Warren
- Johnson, Walter
- Langley, David R
- Li, Aixin
- Li, Jianqing
- Liu, Peiying
- Mastalerz, Harold
- Mathur, Arvind
- Menard, Krista
- Patel, Karishma
- Sack, John
- Sang, Xiaopeng
- Saulnier, Mark
- Smith, Daniel
- Stefanski, Kevin
- Trainor, George
- Velaparthi, Upender
- Zhang, Guifen
- Zimmermann, Kurt
- Vyas, Dolatrai M
Producer: 20091231
In:
Journal of medicinal chemistry vol. 52
Availability: No items available.
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