Results
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1.
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Discovery of potent, selective 4-fluoroproline-based thrombin inhibitors with improved metabolic stability. [electronic resource] by
- Staas, Donnette D
- Savage, Kelly L
- Sherman, Vanessa L
- Shimp, Heidi L
- Lyle, Terry A
- Tran, Lekhanh O
- Wiscount, Catherine M
- McMasters, Daniel R
- Sanderson, Philip E J
- Williams, Peter D
- Lucas, Bobby J
- Krueger, Julie A
- Lewis, S Dale
- White, Rebecca B
- Yu, Sean
- Wong, Bradley K
- Kochansky, Christopher J
- Anari, M Reza
- Yan, Youwei
- Vacca, Joseph P
Producer: 20061124
In:
Bioorganic & medicinal chemistry vol. 14
Availability: No items available.
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2.
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10-Hydroxy-7,8-dihydropyrazino[1',2':1,5]pyrrolo[2,3-d]pyridazine-1,9(2H,6H)-diones: potent, orally bioavailable HIV-1 integrase strand-transfer inhibitors with activity against integrase mutants. [electronic resource] by
- Wiscount, Catherine M
- Williams, Peter D
- Tran, Lekhanh O
- Embrey, Mark W
- Fisher, Thorsten E
- Sherman, Vanessa
- Homnick, Carl F
- Donnette Staas, D
- Lyle, Terry A
- Wai, John S
- Vacca, Joseph P
- Wang, ZiQiang
- Felock, Peter J
- Stillmock, Kara A
- Witmer, Marc V
- Miller, Michael D
- Hazuda, Daria J
- Day, Alysha M
- Gabryelski, Lori J
- Ecto, Linda T
- Schleif, William A
- DiStefano, Daniel J
- Kochansky, Christopher J
- Anari, M Reza
Producer: 20081124
In:
Bioorganic & medicinal chemistry letters vol. 18
Availability: No items available.
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3.
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Design and Synthesis of Piperazine Sulfonamide Cores Leading to Highly Potent HIV-1 Protease Inhibitors. [electronic resource] by
- Bungard, Christopher J
- Williams, Peter D
- Schulz, Jurgen
- Wiscount, Catherine M
- Holloway, M Katharine
- Loughran, H Marie
- Manikowski, Jesse J
- Su, Hua-Poo
- Bennett, David J
- Chang, Lehua
- Chu, Xin-Jie
- Crespo, Alejandro
- Dwyer, Michael P
- Keertikar, Kartik
- Morriello, Gregori J
- Stamford, Andrew W
- Waddell, Sherman T
- Zhong, Bin
- Hu, Bin
- Ji, Tao
- Diamond, Tracy L
- Bahnck-Teets, Carolyn
- Carroll, Steven S
- Fay, John F
- Min, Xu
- Morris, William
- Ballard, Jeanine E
- Miller, Michael D
- McCauley, John A
Publication details: ACS medicinal chemistry letters Dec 2017
In:
ACS medicinal chemistry letters vol. 8
Availability: No items available.
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4.
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Discovery of MK-8718, an HIV Protease Inhibitor Containing a Novel Morpholine Aspartate Binding Group. [electronic resource] by
- Bungard, Christopher J
- Williams, Peter D
- Ballard, Jeanine E
- Bennett, David J
- Beaulieu, Christian
- Bahnck-Teets, Carolyn
- Carroll, Steve S
- Chang, Ronald K
- Dubost, David C
- Fay, John F
- Diamond, Tracy L
- Greshock, Thomas J
- Hao, Li
- Holloway, M Katharine
- Felock, Peter J
- Gesell, Jennifer J
- Su, Hua-Poo
- Manikowski, Jesse J
- McKay, Daniel J
- Miller, Mike
- Min, Xu
- Molinaro, Carmela
- Moradei, Oscar M
- Nantermet, Philippe G
- Nadeau, Christian
- Sanchez, Rosa I
- Satyanarayana, Tummanapalli
- Shipe, William D
- Singh, Sanjay K
- Truong, Vouy Linh
- Vijayasaradhi, Sivalenka
- Wiscount, Catherine M
- Vacca, Joseph P
- Crane, Sheldon N
- McCauley, John A
Producer: 20160720
In:
ACS medicinal chemistry letters vol. 7
Availability: No items available.
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